SCHEMBL7834969

SCHEMBL7834969

CCOC(=O)CC(NC(=O)CNC(=O)c1cc(NC(=N)N)ccc1O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.37
TP53 P04637 1/20 0.37
THRB P10828 1/20 0.37
MEN1 O00255 1/20 0.36
HPGD P15428 1/20 0.36
ITGB3 P05106 2/20 0.35
ITGA2B P08514 1/20 0.35
FADS1 O60427 1/20 0.35
F7 P08709 4/20 0.35
GPR139 Q6DWJ6 2/20 0.35
ALDH1A1 P00352 1/20 0.34
ANO1 Q5XXA6 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
F2 P00734 1/20 0.34
F10 P00742 1/20 0.34
PLAU P00749 1/20 0.34
PLAT P00750 1/20 0.34
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6779352 0.88 ITGB3 (0.41) ITGB3ITGA2BGPR139ITGB1ITGAV
SCHEMBL7346866 0.85 GPR139 (0.41) KMT2ATP53THRBMEN1ITGB3
SCHEMBL7823466 0.83 GPR139 (0.40) TP53THRBITGB3ITGA2BF7
SCHEMBL7339440 0.82 GPR139 (0.41) KMT2ATP53THRBMEN1ITGB3
SCHEMBL6778040 0.81 GPR139 (0.41) KMT2AMEN1HPGDITGB3ITGA2B
SCHEMBL7341087 0.80 GPR139 (0.48) KMT2ATHRBMEN1ITGB3F7
SCHEMBL14450496 0.79 PTGDR2 (0.44) ITGB3ITGA2BALDH1A1POLB
SCHEMBL7835622 0.79 ITGB3 (0.42) KMT2AMEN1ITGB3F7GPR139
SCHEMBL6778730 0.77 ITGB3 (0.40) KMT2AMEN1ITGB3GPR139ITGB1
SCHEMBL7341726 0.77 GPR139 (0.42) KMT2AMEN1ITGB3F7GPR139

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-B1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS SEARLE & CO (US) 2001-07-18 EP claimed