SCHEMBL7835879

SCHEMBL7835879

Nc1nc(C2CC(Br)Cc3ccccc32)nc2nc[nH]c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.40
GDA Q9Y2T3 1/20 0.40
POLA1 P09884 1/20 0.32
LMNA P02545 3/20 0.32
PI4KA P42356 2/20 0.32
PI4K2B Q8TCG2 2/20 0.32
PI4K2A Q9BTU6 2/20 0.32
PI4KB Q9UBF8 2/20 0.32
DRD3 P35462 1/20 0.32
XDH P47989 1/20 0.32
LRRK2 Q5S007 1/20 0.32
PIN1 Q13526 3/20 0.32
CDK1 P06493 3/20 0.32
BRAF P15056 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 2/20 0.32
CCNB1 P14635 2/20 0.32
CCNA2 P20248 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7836200 0.99 PDPK1 (0.39) PDPK1GDAPOLA1LMNAPI4KA
SCHEMBL7830380 0.79 ADRA1A (0.50) PDPK1GDACDK1CYP2D6CCNB1
Hydrochloric Acid SCHEMBL7832458 0.78 ADRA1A (0.49) PDPK1GDAPI4KAPI4K2BPI4K2A
SCHEMBL28984638 0.67 PDPK1 (0.58) PDPK1GDAPOLA1LMNAPI4KA
SCHEMBL7821765 0.66 CDC7 (0.46) PDPK1LMNACDK1CDK2TSHR
SCHEMBL7821652 0.66 CDC7 (0.43) LMNACYP1A2TSHRHSD17B10PKM
SCHEMBL7822155 0.66 LMNA (0.40) LMNACYP1A2CYP2D6CDK2TSHR
SCHEMBL17800816 0.65 PDPK1 (0.54) PDPK1GDAPOLA1LMNAPI4KA
SCHEMBL28482150 0.65 PDPK1 (0.54) PDPK1GDAPOLA1LMNAPI4KA
SCHEMBL3245638 0.64 PDPK1 (0.53) PDPK1GDALMNAPI4KAPI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP claimed
EP-0802914-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.p.A. (IT) 1997-10-29 EP claimed
WO-1997018212-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.P.A. (IT) 1997-05-22 WO claimed
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP disclosed
EP-0802914-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.p.A. (IT) 1997-10-29 EP disclosed
WO-1997018212-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.P.A. (IT) 1997-05-22 WO disclosed