SCHEMBL7835910

SCHEMBL7835910

CCOC(=O)c1nc(C2Cc3c(C(=O)Nc4ccccc4)cccc3C2=O)c[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
RAB9A P51151 3/20 0.40
POLB P06746 1/20 0.40
PKM P14618 1/20 0.40
SMN1; SMN2 Q16637 5/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
GAA P10253 3/20 0.39
NPC1 O15118 2/20 0.39
EPHX2 P34913 1/20 0.39
PTPN11 Q06124 2/20 0.38
JAK3 P52333 2/20 0.38
LMNA P02545 1/20 0.37
TP53 P04637 2/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
HPGD P15428 1/20 0.36
JAK2 O60674 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7847145 0.85 JAK3 (0.34) ALDH1A1POLBPKMMEN1KMT2A
SCHEMBL7846412 0.82 JAK3 (0.34) ALDH1A1MEN1KMT2AGAAJAK3
SCHEMBL7845975 0.72 ROCK2 (0.43) ALDH1A1MEN1KMT2AGAAEPHX2
SCHEMBL7835902 0.71 F2R (0.40) ALDH1A1RAB9APOLBPKMSMN1; SMN2
SCHEMBL7847297 0.68 CYP3A4 (0.51) ALDH1A1MEN1KMT2ALMNATP53
SCHEMBL8098023 0.67 NSD2 (0.39) ALDH1A1POLBMEN1KMT2AGAA
SCHEMBL4884328 0.64 SMN1; SMN2 (0.51) ALDH1A1RAB9APOLBSMN1; SMN2GAA
SCHEMBL10906349 0.63 KDM4E (0.66) ALDH1A1RAB9APOLBPKMSMN1; SMN2
SCHEMBL14823373 0.62 RAB9A (0.58) ALDH1A1RAB9APOLBPKMSMN1; SMN2
SCHEMBL15247066 0.61 RAB9A (0.54) ALDH1A1RAB9APOLBPKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820455-B1 5H, 10H-IMIDAZO [1,2-a]INDENO [1,2-e]PYRAZIN-4-ONE DERIVATIVES, PREPARATION THEREOF, AND DRUGS CONTAINING SAID DERIVATIVES AVENTIS PHARMA SA (FR) 2001-10-31 EP disclosed
US-6057454-A USEFUL FOR TREATING OR PREVENTING ALL ISCHAEMIAS (SUCH AS FOCAL OR GLOBAL ISCHAEMIA) RESULTING FROM CEREBROVASCULAR DISORDERS RHONE-POULENC RORER S.A. (FR) 2000-05-02 US disclosed
US-5902803-A 5H,10H-imidazo 1,2-a!indeno 1,2-e!pyrazin-4-one derivatives, preparation thereof, and drugs containing said derivatives RHONE-POULENC RORER S.A. (FR) 1999-05-11 US disclosed
EP-0820455-A1 5H, 10H-IMIDAZO [1,2-a]INDENO [1,2-e]PYRAZIN-4-ONE DERIVATIVES, PREPARATION THEREOF, AND DRUGS CONTAINING SAID DERIVATIVES Aventis Pharma S.A. (FR) 1998-01-28 EP disclosed
WO-1996031511-A1 5H,10H-IMIDAZO[1,2-a]INDENO[1,2-e]PYRAZIN-4-ONE DERIVATIVES, PREPARATION THEREOF, AND DRUGS CONTAINING SAID DERIVATIVES RHONE-POULENC RORER S.A. (FR) 1996-10-10 WO disclosed