SCHEMBL7836451

SCHEMBL7836451

COc1c(O)ccc2c(C=O)c[nH]c12

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MAPT P10636 1/20 0.48
TRIM24 O15164 2/20 0.47
TRIM33 Q9UPN9 2/20 0.47
PIM3 Q86V86 9/20 0.47
PIM1 P11309 7/20 0.47
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
PIM2 Q9P1W9 2/20 0.43
ERN1 O75460 2/20 0.42
PPARG P37231 1/20 0.42
MAOA P21397 1/20 0.39
TYR P14679 1/20 0.39
CYP2A6 P11509 2/20 0.38
IMPDH2 P12268 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7835597 0.83 ALDH1A1 (0.49) ALDH1A1KDM4EMAPTTRIM24TRIM33
SCHEMBL29952386 0.81 PIM3 (0.51) CA1CA2ALDH1A1KDM4EMAPT
SCHEMBL29958402 0.81 ALDH1A1 (0.48) CA1CA2ALDH1A1KDM4EMAPT
SCHEMBL29955110 0.81 ALDH1A1 (0.48) CA1CA2ALDH1A1KDM4EMAPT
SCHEMBL29954723 0.76 PIM3 (0.51) ALDH1A1KDM4EMAPTTRIM24TRIM33
SCHEMBL29952798 0.76 PIM3 (0.50) ALDH1A1KDM4EMAPTTRIM24TRIM33
SCHEMBL29957633 0.76 TRIM24 (0.47) ALDH1A1KDM4EMAPTTRIM24TRIM33
SCHEMBL14519078 0.75 PIM3 (0.65) ALDH1A1KDM4EMAPTTRIM24TRIM33
SCHEMBL7836770 0.75 TUBB1 (0.57)
SCHEMBL29955386 0.73 TRIM24 (0.66) CA1CA2TRIM24TRIM33PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0680950-B1 PROPENONE DERIVATIVES KYOWA HAKKO KOGYO KK (JP) 2001-05-23 EP disclosed
US-5952355-A 1-ETHER-SUBSTITUTED PHENYL-3-INDOL-3-YL-2-PROPEN-1-ONE DERIVATIVES; ANTITUMOR AND -CARCINOGENIC AGENTS; IMMUNOSUPPRESSANTS; AUTOIMMUNE DISEASES; SIDE EFFECT REDUCTION KYOWA HAKKO KOGYO CO., LTD. (JP) 1999-09-14 US disclosed
EP-0680950-A1 PROPENONE DERIVATIVE KYOWA HAKKO KOGYO CO., LTD. (JP) 1995-11-08 EP disclosed