SCHEMBL7837474

SCHEMBL7837474

COc1ccc(-c2ccc3c(c2)NC(=O)/C3=C\c2[nH]c3c(c2C)CCCC3)cc1

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 14/20 0.71
KDR P35968 13/20 0.71
FGFR1 P11362 12/20 0.71
SRC P12931 7/20 0.71
EGFR P00533 3/20 0.61
CHEK1 O14757 2/20 0.50
KIT P10721 1/20 0.47
FLT4 P35916 1/20 0.47
FLT3 P36888 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7837476 1.00 PDGFRB (0.71) PDGFRBKDRFGFR1SRCEGFR
SCHEMBL8205880 0.92 PDGFRB (0.72) PDGFRBKDRFGFR1SRCEGFR
SCHEMBL8205878 0.92 PDGFRB (0.72) PDGFRBKDRFGFR1SRCEGFR
SCHEMBL8211103 0.86 PDGFRB (0.72) PDGFRBKDRFGFR1SRCEGFR
SCHEMBL7825508 0.86 PDGFRB (0.72) PDGFRBKDRFGFR1SRCEGFR
SCHEMBL6393305 0.83 FGFR1 (1.00) PDGFRBKDRFGFR1SRCEGFR
SCHEMBL6393309 0.83 FGFR1 (1.00) PDGFRBKDRFGFR1SRCEGFR
SCHEMBL6701476 0.77 SRC (0.78) PDGFRBKDRFGFR1SRCEGFR
SCHEMBL6391952 0.76 FGFR1 (1.00) PDGFRBKDRFGFR1SRCEGFR
SCHEMBL6391950 0.76 FGFR1 (1.00) PDGFRBKDRFGFR1SRCEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1066257-A2 HETEROCYLIC CLASSES OF COMPOUNDS FOR THE MODULATING TYROSINE PROTEIN KINASE Sugen, Inc. (US) 2001-01-10 EP disclosed
WO-1999048868-A2 HETEROCYCLIC CLASSES OF COMPOUNDS FOR THE MODULATING TYROSINE PROTEIN KINASE SUGEN, INC. (US) 1999-09-30 WO disclosed