SCHEMBL7839166

SCHEMBL7839166

COC(=O)c1c(C)[nH]c2c(-c3cccc(C)n3)cccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 3/20 0.51
LMNA P02545 4/20 0.43
GAA P10253 2/20 0.43
HTT P42858 2/20 0.43
TSHR P16473 1/20 0.43
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
ALDH1A1 P00352 5/20 0.38
MAPT P10636 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX5 P09917 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KDM4E B2RXH2 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7218658 0.75 NR4A2 (0.59) NR4A2LMNAGAAHTTTSHR
SCHEMBL7839279 0.75 NR4A2 (0.59) NR4A2LMNAGAAHTTTSHR
SCHEMBL5237030 0.75 NR4A2 (0.59) NR4A2LMNAGAAHTTTSHR
SCHEMBL29217694 0.72 NR4A2 (0.43) NR4A2LMNAGAAHTTTSHR
SCHEMBL20842473 0.70 TGFBR1 (0.49) TSHRKMT2AMEN1KDM4ECCR1
SCHEMBL29163735 0.70 L3MBTL1 (0.52) KMT2AMEN1ALDH1A1KDM4ECCR1
SCHEMBL16502656 0.70 TGFBR1 (0.46) LMNAGAAHTTKMT2AMEN1
SCHEMBL7839162 0.70 NR4A2 (0.49) NR4A2LMNAKMT2AMEN1MAPT
SCHEMBL10717437 0.69 HTT (0.67) NR4A2LMNAGAAHTTTSHR
SCHEMBL28490176 0.69 KDM4E (0.45) LMNAHTTKMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140946-A2 QUINOLINE DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 2001-10-10 EP disclosed
WO-2000035919-A2 QUINOLINE DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 2000-06-22 WO disclosed