SCHEMBL7840281

SCHEMBL7840281

O=C(O)Cc1ccc(O)c2[nH]c(=O)sc12

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 15/20 0.47
ADRB1 P08588 5/20 0.47
ABCB11 O95342 2/20 0.42
DRD2 P14416 1/20 0.42
PDE4A P27815 1/20 0.42
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13225820 0.83 CYP1A2 (0.44) ADRB2ADRB1GRIN2DGRIN3BGRIN1
SCHEMBL12119358 0.82 ADRB2 (0.54) ADRB2ADRB1
SCHEMBL4555603 0.81 ADRB2 (0.49) ADRB2ADRB1ABCB11DRD2PDE4A
SCHEMBL4440137 0.79 ADRB2 (0.56) ADRB2ADRB1ABCB11DRD2PDE4A
Acetic Acid SCHEMBL4742751 0.79 ADRB2 (0.47) ADRB2ADRB1ABCB11DRD2PDE4A
SCHEMBL14291843 0.78 ADRB2 (0.52) ADRB2ADRB1
SCHEMBL4740762 0.78 ADRB2 (0.52) ADRB2ADRB1ABCB11DRD2PDE4A
SCHEMBL4788200 0.78 ADRB2 (0.47) ADRB2ADRB1ABCB11DRD2PDE4A
Bromide SCHEMBL1683003 0.77 ADRB2 (0.51) ADRB2ADRB1ABCB11DRD2PDE4A
SCHEMBL4715369 0.77 ADRB2 (0.46) ADRB2ADRB1ABCB11DRD2PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0558677-B1 BIOLOGICALLY ACTIVE AMINES ASTRAZENECA AB (SE) 2001-08-16 EP disclosed
US-5763465-A 7-(2-aminoethyl) benzothiazolones ASTRA PHARMACEUTICALS LIMITED (GB) 1998-06-09 US disclosed
US-5648370-A 7-(2-aminoethyl) benzothiazolones ASTRA PHARMACEUTICALS LIMITED (GB) 1997-07-15 US disclosed
WO-1993023385-A1 BIOLOGICALLY ACTIVE AMINES FISONS PLC (GB) 1993-11-25 WO disclosed
EP-0558677-A1 BIOLOGICALLY ACTIVE AMINES Astra Pharmaceuticals Limited (GB) 1993-09-08 EP disclosed
WO-1992008708-A1 BIOLOGICALLY ACTIVE AMINES FISONS PLC (GB) 1992-05-29 WO disclosed