SCHEMBL7840451

SCHEMBL7840451

COc1ccc2cc(C(Oc3c[nH]cn3)c3ccncc3)ccc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.40
ABCB11 O95342 1/20 0.37
PDGFRB P09619 2/20 0.37
PDGFRA P16234 2/20 0.37
RIOK2 Q9BVS4 4/20 0.37
AKR1C3 P42330 4/20 0.36
AKR1C2 P52895 4/20 0.36
PTGS2 P35354 3/20 0.36
PTGS1 P23219 2/20 0.36
TSHR P16473 2/20 0.36
CDC42 P60953 1/20 0.36
RAC1 P63000 1/20 0.36
CYP1A2 P05177 1/20 0.36
SLC22A6 Q4U2R8 1/20 0.36
ALOX5 P09917 1/20 0.36
RAB9A P51151 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
GSK3A P49840 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7846759 0.86 CYP11B2 (0.43) CYP17A1CYP1A2RAB9AMAPTCYP2C9
SCHEMBL5752670 0.75 ABCB11 (0.42) ABCB11RIOK2AKR1C3AKR1C2PTGS2
SCHEMBL5750067 0.72 ABCB11 (0.43) ABCB11RIOK2AKR1C3AKR1C2PTGS2
SCHEMBL5750801 0.69 ABCB11 (0.51) CYP17A1ABCB11RIOK2AKR1C3AKR1C2
SCHEMBL7840454 0.69 RIOK2 (0.41) ABCB11RIOK2AKR1C3AKR1C2PTGS2
SCHEMBL4828425 0.66 AKR1C3 (0.54) ABCB11RIOK2AKR1C3AKR1C2PTGS2
SCHEMBL4828431 0.66 AKR1C3 (0.47) CYP17A1ABCB11RIOK2AKR1C3AKR1C2
SCHEMBL7806036 0.64 ABCB11 (0.46) CYP17A1ABCB11RIOK2AKR1C3AKR1C2
SCHEMBL5751571 0.64 CYP17A1 (0.45) CYP17A1PDGFRBPDGFRACYP1A2
SCHEMBL31546885 0.64 NPC1 (0.53) CYP17A1CYP1A2RAB9ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1073640-A1 NAPHTHALENE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2001-02-07 EP disclosed
WO-1999054309-A1 NAPHTHALENE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-10-28 WO disclosed