SCHEMBL7840744

SCHEMBL7840744

COc1ccc(CCNC(=O)CCSCC(=O)NCCc2ccccc2)c2sc(=O)[nH]c12

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 7/20 0.51
ALDH1A1 P00352 2/20 0.46
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TAAR1 Q96RJ0 1/20 0.44
HSD17B10 Q99714 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.42
USP2 O75604 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7829366 0.83 ADRB2 (0.51) ADRB2HTTTAAR1HSD17B10CYP1A2
SCHEMBL7839860 0.81 SMN1; SMN2 (0.46) ALDH1A1LMNAHTTSMN1; SMN2TAAR1
SCHEMBL8532601 0.77 ADRB2 (0.75) ADRB2
SCHEMBL10499469 0.77 KMT2A (0.66) ALDH1A1LMNAHTTSMN1; SMN2HSD17B10
SCHEMBL10452367 0.77 KMT2A (0.66) ALDH1A1LMNAHTTSMN1; SMN2HSD17B10
SCHEMBL8673879 0.77 ADRB2 (0.53) ADRB2
SCHEMBL8532543 0.77 ADRB2 (0.69) ADRB2
SCHEMBL7295271 0.72 SLC2A1 (0.61) ALDH1A1KDM4EHPGD
SCHEMBL8671939 0.72 ADRB2 (0.51) ADRB2
Hydrochloric Acid SCHEMBL8899662 0.71 ADRB2 (0.63) ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0558677-B1 BIOLOGICALLY ACTIVE AMINES ASTRAZENECA AB (SE) 2001-08-16 EP disclosed
US-5763465-A 7-(2-aminoethyl) benzothiazolones ASTRA PHARMACEUTICALS LIMITED (GB) 1998-06-09 US disclosed
US-5648370-A 7-(2-aminoethyl) benzothiazolones ASTRA PHARMACEUTICALS LIMITED (GB) 1997-07-15 US disclosed