SCHEMBL7841767

SCHEMBL7841767

C[C@H]1C=C[C@@H](N)[C@H]2CN(c3ncc4c(=O)c(C(=O)O)cn(C5CC5)c4c3F)C[C@H]21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 7/20 0.44
TOP2B Q02880 7/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
KCNH2 Q12809 4/20 0.43
POLB P06746 3/20 0.43
CACNA1F O60840 1/20 0.43
MAPK1 P28482 1/20 0.43
CACNA1D Q01668 1/20 0.43
CACNA1S Q13698 1/20 0.43
CACNA1C Q13936 1/20 0.43
ALDH1A1 P00352 2/20 0.42
OPRM1 P35372 2/20 0.42
CHRM2 P08172 1/20 0.42
CHRM1 P11229 1/20 0.42
OPRD1 P41143 1/20 0.42
DPP4 P27487 5/20 0.41
KDM4E B2RXH2 1/20 0.40
PRKD3 O94806 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7850903 0.90 POLB (0.46) TOP2ATOP2BMEN1KMT2AKCNH2
SCHEMBL7841774 0.89 TOP2A (0.33) TOP2ATOP2BMEN1KMT2AKCNH2
Hydrochloric Acid SCHEMBL8697994 0.89 POLB (0.45) TOP2ATOP2BMEN1KMT2AKCNH2
Bromide SCHEMBL8692350 0.89 POLB (0.45) TOP2ATOP2BMEN1KMT2AKCNH2
SCHEMBL7853917 0.85 TOP2A (0.42) TOP2ATOP2BMEN1KMT2AKCNH2
SCHEMBL9145431 0.84 KCNH2 (0.47) TOP2ATOP2BMEN1KMT2AKCNH2
SCHEMBL8133384 0.84 ALDH1A1 (0.56) TOP2ATOP2BMEN1KMT2AKCNH2
Hydrochloric Acid SCHEMBL9149906 0.83 KCNH2 (0.47) TOP2ATOP2BMEN1KMT2AKCNH2
SCHEMBL7841768 0.81 EPHA2 (0.56) TOP2ATOP2BMEN1KMT2APOLB
SCHEMBL7851044 0.81 KDM4E (0.42) TOP2ATOP2BKCNH2POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726270-B1 Derivatives of 1,6-naphthyridone carboxylic acids BAYER AG (DE) 2001-05-23 EP disclosed
US-5811433-A ANTIMICROBIALS BAYER AKTIENGESELLSCHAFT (DE) 1998-09-22 US disclosed
EP-0726270-A1 Derivatives of 1,6-naphthyridine carboxylic acids BAYER AG (DE) 1996-08-14 EP disclosed