SCHEMBL7841891

SCHEMBL7841891

O=[N+]([O-])c1cccnc1-c1ncccn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.55
POLB P06746 1/20 0.53
ALDH1A1 P00352 6/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2C9 P11712 2/20 0.49
NCOA1 Q15788 1/20 0.49
NCOA3 Q9Y6Q9 1/20 0.49
CYP2C19 P33261 1/20 0.49
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
RAB9A P51151 2/20 0.47
TRPV1 Q8NER1 1/20 0.47
PKM P14618 1/20 0.45
LMNA P02545 3/20 0.45
PAX8 Q06710 1/20 0.45
MAPT P10636 4/20 0.45
KDM4E B2RXH2 2/20 0.45
CTSB P07858 2/20 0.45
GAA P10253 1/20 0.45
IDO1 P14902 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29940575 0.90 PDE10A (0.60) PDE10APOLBALDH1A1CYP1A2CYP2C9
SCHEMBL6512953 0.90 PDE10A (0.60) PDE10APOLBALDH1A1CYP1A2CYP2C9
SCHEMBL30794281 0.86 PDE10A (0.46) PDE10APOLBALDH1A1CYP1A2CYP2C9
SCHEMBL444703 0.85 ALDH1A1 (0.53) PDE10APOLBALDH1A1CYP1A2CYP2C9
SCHEMBL28567279 0.83 PDE10A (0.50) PDE10APOLBALDH1A1CYP1A2CYP2C9
SCHEMBL1736457 0.80 PAX8 (0.57) PDE10APOLBALDH1A1CYP1A2CYP2C9
SCHEMBL1736168 0.80 MEN1 (0.57) PDE10APOLBALDH1A1CYP1A2CYP2C9
SCHEMBL1738384 0.80 MAPT (0.52) PDE10APOLBALDH1A1CYP1A2CYP2C9
SCHEMBL30269976 0.80 CYP2A6 (0.54) PDE10APOLBALDH1A1CYP1A2CYP2C9
SCHEMBL27930436 0.80 TRPV1 (0.51) PDE10APOLBALDH1A1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150955-A2 G-PROTEIN COUPLED HEPTAHELICAL RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF Millennium Pharmaceuticals, Inc. (US) 2001-11-07 EP disclosed
WO-2000046203-A2 G-PROTEIN COUPLED HEPTAHELICAL RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2000-08-10 WO disclosed