SCHEMBL7841944

SCHEMBL7841944

COCC(Cc1ccccc1)S(=O)(=O)Nc1nn(CCOC(C)=O)c(OC)c1-c1ccc2c(c1)OCO2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
CYP19A1 P11511 1/20 0.37
MAPK1 P28482 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
SCD5 Q86SK9 1/20 0.37
EDNRB P24530 7/20 0.37
EDNRA P25101 6/20 0.37
ALDH1A1 P00352 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
HPGD P15428 2/20 0.36
CYP2C19 P33261 2/20 0.36
TP53 P04637 2/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
GAA P10253 1/20 0.36
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ITGB1 P05556 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6293272 0.76 EDNRB (0.40) CYP19A1MAPK1NPSR1SCD5EDNRB
SCHEMBL6288916 0.76 TSHR (0.41) TSHRCYP19A1MAPK1NPSR1SCD5
SCHEMBL6289705 0.66 CYP19A1 (0.49) TSHRCYP19A1MAPK1NPSR1SCD5
SCHEMBL6289234 0.62 RIPK2 (0.44) TSHRMAPK1EDNRBEDNRAALDH1A1
SCHEMBL7216623 0.61 CYP19A1 (0.42) CYP19A1MAPK1NPSR1SCD5EDNRB
SCHEMBL6289617 0.61 CYP1A2 (0.50) CYP19A1MAPK1NPSR1SCD5EDNRB
SCHEMBL6289186 0.60 LMNA (0.50) CYP19A1MAPK1NPSR1SCD5EDNRB
SCHEMBL6289188 0.60 LMNA (0.50) CYP19A1MAPK1NPSR1SCD5EDNRB
SCHEMBL20610727 0.60 CYP3A4 (0.75) TSHREDNRAALDH1A1HPGDTP53
SCHEMBL30133684 0.60 CAPN1 (0.50) ALDH1A1GAAITGB1ITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1072597-A1 Pyrazoles and their use as endothelin antagonists Pfizer Limited (GB) 2001-01-31 EP disclosed