SCHEMBL7841970

SCHEMBL7841970

COc1ccnc(-c2cc(NC(=NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)ccc2C)c1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 15/20 0.36
BRAF P15056 15/20 0.36
KDM4C Q9H3R0 2/20 0.35
KDM6B O15054 1/20 0.35
KDM5A P29375 1/20 0.35
KDM4D Q6B0I6 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
KDM2A Q9Y2K7 1/20 0.35
KDM3A Q9Y4C1 1/20 0.35
DYRK1A Q13627 1/20 0.35
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
CCR8 P51685 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7240473 0.87 CCR1 (0.33) KDM4CKDM6BKDM5AKDM4DKDM5B
SCHEMBL7843005 0.85 CYP17A1 (0.41) BRAF
SCHEMBL7853175 0.84 KDM4E (0.40) DYRK1ACCR1CCR5CCR8
SCHEMBL7238742 0.82 CCR1 (0.38) DYRK1ACCR1CCR5CCR8
SCHEMBL3778074 0.78 POLB (0.43) RAF1
SCHEMBL3778070 0.78 POLB (0.43) RAF1
SCHEMBL13785800 0.78 POLB (0.43) RAF1
SCHEMBL7845048 0.78 KDR (0.41)
SCHEMBL7846741 0.78 AAK1 (0.38) CCR1CCR5CCR8
SCHEMBL17560319 0.78 RAB9A (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed