SCHEMBL7843005

SCHEMBL7843005

COc1ccnc(-c2cccc(NC(=NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.41
MAPT P10636 4/20 0.40
POLB P06746 3/20 0.40
TP53 P04637 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
BRAF P15056 4/20 0.40
FYN P06241 2/20 0.39
CNR1 P21554 1/20 0.39
GRM4 Q14833 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
MAPKAPK2 P49137 1/20 0.38
KDR P35968 1/20 0.38
HDAC3 O15379 2/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC2 Q92769 2/20 0.38
HDAC10 Q969S8 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7847281 0.91 KMT2A (0.41) CYP17A1MAPTPOLBMEN1KMT2A
SCHEMBL7846551 0.88 CNR1 (0.52) CYP17A1MAPTTP53MEN1KMT2A
SCHEMBL17560319 0.86 RAB9A (0.48) MAPTPOLBTP53MEN1KMT2A
SCHEMBL7841970 0.85 RAF1 (0.36) BRAF
SCHEMBL7845384 0.84 MAPT (0.43) CYP17A1MAPTPOLBMEN1KMT2A
SCHEMBL7853175 0.84 KDM4E (0.40) MAPTPOLBTP53
SCHEMBL7845048 0.83 KDR (0.41) KDR
SCHEMBL7846741 0.83 AAK1 (0.38) TP53CYP1A2CYP3A4CYP2C19
SCHEMBL7240473 0.81 CCR1 (0.33) KDR
SCHEMBL7229573 0.81 CCR1 (0.40) MAPTTP53MAPKAPK2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed