SCHEMBL7842311

SCHEMBL7842311

N#Cc1c(Cn2ccnn2)nc2ccccc2c1Nc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 8/20 0.46
CYP19A1 P11511 4/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 1/20 0.40
RAD52 P43351 4/20 0.40
KMT2A Q03164 4/20 0.40
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
POLB P06746 3/20 0.37
TOP2A P11388 1/20 0.37
TOP2B Q02880 1/20 0.37
MAPT P10636 1/20 0.37
OPRM1 P35372 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7836868 0.84 KDM1A (0.43) KDM1AKDM4EALDH1A1RAD52KMT2A
SCHEMBL7845566 0.81 KDM1A (0.47) KDM1AKDM4EALDH1A1RAD52KMT2A
SCHEMBL6071828 0.81 CYP19A1 (0.44) CYP19A1KDM4EALDH1A1RAD52KMT2A
SCHEMBL7842318 0.80 MEN1 (0.47) KDM1ACYP19A1KDM4EALDH1A1KMT2A
SCHEMBL7999974 0.80 KDM1A (0.43) KDM1AKDM4EALDH1A1RAD52KMT2A
SCHEMBL6071833 0.73 CYP19A1 (0.46) CYP19A1KDM4EALDH1A1RAD52KMT2A
SCHEMBL7689595 0.70 KDM1A (0.57) KDM1AKDM4EALDH1A1RAD52KMT2A
SCHEMBL7826829 0.69 KDM1A (0.43) KDM1AKDM4EALDH1A1RAD52KMT2A
SCHEMBL4557943 0.68 KDM1A (0.47) KDM1AKDM4EALDH1A1RAD52KMT2A
SCHEMBL28613370 0.67 KDM1A (0.49) KDM1AKDM4EALDH1A1RAD52KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117659-A1 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS American Cyanamid Company (US) 2001-07-25 EP disclosed
WO-2000018761-A1 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS AMERICAN CYANAMID COMPANY (US) 2000-04-06 WO disclosed