SCHEMBL7999974

SCHEMBL7999974

N#Cc1c(Cn2ncnn2)nc2ccccc2c1Nc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 6/20 0.43
KMT2A Q03164 3/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 2/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ABCG2 Q9UNQ0 3/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
RAF1 P04049 1/20 0.35
MAP2K1 Q02750 1/20 0.35
POLB P06746 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HDAC3 O15379 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7845566 0.86 KDM1A (0.47) KDM1AKMT2AKDM4EALDH1A1MEN1
SCHEMBL7836868 0.80 KDM1A (0.43) KDM1AKMT2AKDM4EALDH1A1MEN1
SCHEMBL7842311 0.80 KDM1A (0.46) KDM1AKMT2AKDM4EALDH1A1MEN1
SCHEMBL7999981 0.80 MEN1 (0.45) KDM1AKMT2AKDM4EALDH1A1MEN1
SCHEMBL7689595 0.70 KDM1A (0.57) KDM1AKMT2AKDM4EALDH1A1MEN1
SCHEMBL7826829 0.69 KDM1A (0.43) KDM1AKMT2AKDM4EALDH1A1MEN1
SCHEMBL28613370 0.67 KDM1A (0.49) KDM1AKMT2AKDM4EALDH1A1MEN1
SCHEMBL28618474 0.66 ALDH1A1 (0.50) KDM1AKMT2AKDM4EALDH1A1MEN1
SCHEMBL4557943 0.65 KDM1A (0.47) KDM1AKMT2AKDM4EALDH1A1CYP1A2
SCHEMBL7845574 0.65 MEN1 (0.48) KMT2AKDM4EALDH1A1MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288082-B1 COMPOUNDS SUCH AS 6,7-DIETHOXY-4-(INDAN-5-YLAMINO) -QUINOLINE-3-CARBONITRILE USED AS ANTINEOPLASTIC AGENTS AND IN THE TREATMENT OF POLYCYCSTIC KIDNEY DISEASE AMERICAN CYANAMID COMPANY 2001-09-11 US disclosed