SCHEMBL7842318

SCHEMBL7842318

N#Cc1c(Nc2ccccc2)nc2ccccc2c1Cn1ccnn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
NPSR1 Q6W5P4 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
CYP19A1 P11511 4/20 0.41
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 3/20 0.40
LMNA P02545 2/20 0.38
CYP1A2 P05177 2/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ABCG2 Q9UNQ0 5/20 0.37
KDM1A O60341 1/20 0.37
NPY5R Q15761 1/20 0.36
USP2 O75604 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7836872 0.84 MEN1 (0.45) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL6071833 0.82 CYP19A1 (0.46) MEN1KMT2ANPSR1RXFP1CYP19A1
SCHEMBL7845574 0.81 MEN1 (0.48) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL7842311 0.80 KDM1A (0.46) MEN1KMT2ANPSR1CYP19A1ALDH1A1
SCHEMBL7999981 0.80 MEN1 (0.45) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL7999933 0.75 MEN1 (0.51) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL6071828 0.72 CYP19A1 (0.44) KMT2ANPSR1RXFP1CYP19A1ALDH1A1
SCHEMBL20259096 0.70 ALDH1A1 (0.58) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL7689600 0.70 ALDH1A1 (0.51) MEN1KMT2ANPSR1RXFP1ALDH1A1
SCHEMBL7826836 0.69 MEN1 (0.45) MEN1KMT2ANPSR1RXFP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117659-A1 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS American Cyanamid Company (US) 2001-07-25 EP disclosed
WO-2000018761-A1 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS AMERICAN CYANAMID COMPANY (US) 2000-04-06 WO disclosed