SCHEMBL7843083

SCHEMBL7843083

COC(=O)CC1=C(C(=O)O)C(c2c(Cl)cccc2Cl)C(C(=O)O)=C(CCc2ccccc2OC)N1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
NR3C2 P08235 1/20 0.39
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
CNR1 P21554 1/20 0.37
USP2 O75604 1/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6949307 0.89 CYP2C9 (0.32) ALDH1A1NPC1RAB9AKDM4EGAA
SCHEMBL6946876 0.89 TTR (0.35) ALDH1A1NPC1RAB9AUSP2MEN1
SCHEMBL6153461 0.89 CYP4F2 (0.34) ALDH1A1NPC1RAB9AKDM4EUSP2
SCHEMBL6153189 0.88 CYP2C9 (0.32) ALDH1A1NPC1RAB9AKDM4EUSP2
SCHEMBL6153097 0.87 ALDH1A1 (0.31) ALDH1A1NR3C2HPGDHTT
SCHEMBL7836265 0.86 SLC7A5 (0.39) ALDH1A1NPC1RAB9AKDM4EMEN1
SCHEMBL6152821 0.86 KMT2A (0.31) ALDH1A1KDM4EUSP2MEN1KMT2A
SCHEMBL6940682 0.86 PPARD (0.35) ALDH1A1NPC1RAB9AKDM4EMEN1
SCHEMBL7841344 0.86 MAPT (0.35) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL6153144 0.85 PPARG (0.35) ALDH1A1MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777653-B1 DIHYGROPYRIDINE DERIVATIVES AS BRADYKININ ANTAGONISTS PFIZER (US) 2001-08-22 EP disclosed
US-5859011-A Dihydropyridine derivatives as bradykinin antagonist PFIZER INC. (US) 1999-01-12 US disclosed
WO-1996006082-A1 DIHYDROPYRIDINE DERIVATIVES AS BRADYKININ ANTAGONISTS PFIZER INC. (US) 1996-02-29 WO disclosed