SCHEMBL7843461

SCHEMBL7843461

CCCCc1c[nH]c2c(c1=O)CCCC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.39
GABRB2 P47870 1/20 0.39
ALDH1A1 P00352 6/20 0.38
KDM4E B2RXH2 4/20 0.38
HPGD P15428 3/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HIF1A Q16665 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
USP2 O75604 1/20 0.32
ALPL P05186 1/20 0.32
DDB1 Q16531 1/20 0.32
CRBN Q96SW2 1/20 0.32
BRD9 Q9H8M2 1/20 0.32
HTR1A P08908 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6160790 0.70 TSHR (0.44) GABRA1GABRB2ALDH1A1KDM4EHPGD
SCHEMBL6681210 0.70 MPO (0.41) ALDH1A1KDM4ECYP2D6MEN1KMT2A
SCHEMBL6407362 0.70 SLC6A4 (0.45) HTR1A
SCHEMBL6696394 0.69 MAPT (0.32) MAPT
SCHEMBL6697504 0.69 SLC6A4 (0.44) HTR1A
SCHEMBL10551768 0.67 HSD17B10 (0.42) ALDH1A1KDM4ETP53MAPTSMN1; SMN2
SCHEMBL19032105 0.67 ALDH1A1 (0.40) ALDH1A1KDM4EMAPTSMN1; SMN2MEN1
SCHEMBL1369026 0.66 HTR1D (0.43) CYP1A2CYP2D6MAPTSMN1; SMN2HTR1A
SCHEMBL5396500 0.66 MAPT (0.49) MAPTHTR1ALMNA
SCHEMBL2392492 0.66 KDM4E (0.60) GABRA1GABRB2ALDH1A1KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0498723-B1 Nitrogen containing bicycle compounds, method for their preparation, their use as pharmaceutical and compositions containing them AVENTIS PHARMA SA (FR) 2001-09-19 EP disclosed
US-6004979-A ANGIOTENSIN II INHIBITORS; 4-((CARBOXY)ARYLOXY)-QUINOLINE DERIVATIVES HOECHST MARION ROUSSEL (FR) 1999-12-21 US disclosed
US-5985894-A USEFUL IN THE TREATMENT OF CARDIOVASCULAR ILLNESSES HOECHST MARION ROUSSEL (FR) 1999-11-16 US disclosed
US-5817674-A ANTIOTENSIN II RECEPTOR ANTAGONISTS ROUSSEL UCLAF (FR) 1998-10-06 US disclosed