SCHEMBL7843799

SCHEMBL7843799

NCCCN1CCc2cc(F)c(F)cc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 8/20 0.46
HTR2C P28335 7/20 0.46
HTR2B P41595 7/20 0.46
EPHX2 P34913 1/20 0.40
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
CDK4 P11802 1/20 0.38
ALOX15 P16050 1/20 0.38
CCND1 P24385 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
NFKB1 P19838 1/20 0.35
HIF1A Q16665 1/20 0.35
AR P10275 2/20 0.34
CHRM1 P11229 2/20 0.33
CHRM2 P08172 1/20 0.33
CHRM3 P20309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7841495 0.87 HTR2A (0.62) HTR2AHTR2CHTR2BEPHX2ALDH1A1
SCHEMBL7833793 0.82 EPHX2 (0.46) HTR2AEPHX2ALDH1A1MEN1USP2
Ammonia Solution, Strong SCHEMBL906070 0.79 HTR2A (0.46) HTR2AHTR2CHTR2BALDH1A1MEN1
SCHEMBL7674589 0.79 HTR2A (0.58) HTR2AHTR2CHTR2BEPHX2ALDH1A1
SCHEMBL7840357 0.76 ALDH1A1 (0.42) HTR2AHTR2CHTR2BEPHX2ALDH1A1
SCHEMBL7833297 0.75 HTR2A (0.42) HTR2AHTR2CHTR2BEPHX2ALDH1A1
Hydrochloric Acid SCHEMBL7845930 0.74 HTR2A (0.57) HTR2AHTR2CHTR2BEPHX2ALDH1A1
SCHEMBL6216648 0.74 ALDH1A1 (0.72) HTR2AEPHX2ALDH1A1MEN1USP2
SCHEMBL906067 0.73 HTR2A (0.78) HTR2AHTR2CHTR2BCYP1A2CYP3A4
SCHEMBL4572835 0.71 CHRM2 (0.54) HTR2AHTR2CHTR2BALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109784-A1 INDOLINE DERIVATIVES AS 5-HT2B AND/OR 5-HT2C RECEPTOR LIGANDS VERNALIS RESEARCH LIMITED (GB) 2001-06-27 EP claimed
WO-2000012475-A1 INDOLINE DERIVATIVES AS 5-HT2B AND/OR 5-HT2C RECEPTOR LIGANDS VERNALIS RESEARCH LIMITED (GB) 2000-03-09 WO claimed