SCHEMBL7843813

SCHEMBL7843813

CSC(N)=Nc1nc(C)c(-c2cc(C)ccn2)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.39
CCR5 P51681 1/20 0.39
CCR8 P51685 1/20 0.39
PLAU P00749 1/20 0.38
CDK4 P11802 6/20 0.35
CDK2 P24941 6/20 0.35
CCNE1 P24864 1/20 0.35
NR2F2 P24468 1/20 0.35
ATP4A P20648 2/20 0.32
ATP4B P51164 2/20 0.32
MAPT P10636 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP2A6 P11509 1/20 0.31
METAP2 P50579 1/20 0.31
NOS3 P29474 2/20 0.31
NOS1 P29475 2/20 0.31
NOS2 P35228 2/20 0.31
KDM4E B2RXH2 2/20 0.31
PLK1 P53350 2/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7229276 0.87 NOS3 (0.42) CCR1CCR5CCR8PLAUNOS3
Hydrochloric Acid SCHEMBL7231887 0.86 NOS3 (0.42) CCR1CCR5CCR8PLAUNOS3
Hydrochloric Acid SCHEMBL7238267 0.81 CCR1 (0.38) CCR1CCR5CCR8PLAUCDK4
SCHEMBL7238645 0.80 SMN1; SMN2 (0.37) CCR1CCR5CCR8PLAUCDK4
SCHEMBL7239613 0.79 SMN1; SMN2 (0.46) CCR1CCR5CCR8CDK4CDK2
SCHEMBL925682 0.72 CCR1 (0.52) CCR1CCR5CCR8CDK4CDK2
SCHEMBL7229862 0.72 CCR1 (0.41) CCR1CCR5CCR8CDK4CDK2
SCHEMBL7229860 0.72 CCR1 (0.41) CCR1CCR5CCR8CDK4CDK2
SCHEMBL7229076 0.70 PIK3CA (0.40) CCR1CCR5CCR8NR2F2MAPT
SCHEMBL7240097 0.70 PIK3CA (0.40) CCR1CCR5CCR8NR2F2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed