SCHEMBL7843844

SCHEMBL7843844

CC(C)(C)OC(=O)N=C(N)Nc1cccc(-c2ncccc2O[Si](C)(C)C(C)(C)C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.36
CYP17A1 P05093 1/20 0.36
SIRT1 Q96EB6 1/20 0.34
KDM4E B2RXH2 4/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
TRPV1 Q8NER1 1/20 0.33
ALDH1A1 P00352 3/20 0.33
HDAC3 O15379 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC10 Q969S8 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
NPC1 O15118 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
RAB9A P51151 1/20 0.33
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7843692 0.87 TDP2 (0.40) TDP2CYP17A1KDM4ESMN1; SMN2HDAC3
SCHEMBL7846042 0.85 CYP17A1 (0.34) TDP2CYP17A1KDM4ESMN1; SMN2TRPV1
SCHEMBL7843840 0.78 HRH2 (0.34) TDP2KDM4E
SCHEMBL7846853 0.76 CYP17A1 (0.41) TDP2CYP17A1SIRT1KDM4EALDH1A1
SCHEMBL7236713 0.74 NPFFR1 (0.35) TDP2CYP17A1KDM4ETRPV1ALDH1A1
SCHEMBL7230492 0.72 MAP4K4 (0.43) ALDH1A1NPC1POLB
SCHEMBL7841418 0.71 CYP17A1 (0.42) TDP2CYP17A1TRPV1HDAC1NPC1
SCHEMBL7842830 0.70 CYP17A1 (0.41) TDP2CYP17A1KDM4EALDH1A1HDAC3
SCHEMBL23455338 0.70 NPC1 (0.48) SMN1; SMN2ALDH1A1NPC1RAB9APOLB
SCHEMBL30001020 0.70 NPC1 (0.48) SMN1; SMN2ALDH1A1NPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed