SCHEMBL7846853

SCHEMBL7846853

COc1cccnc1-c1cccc(NC(=NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.41
TDP2 O95551 1/20 0.40
ALDH1A1 P00352 2/20 0.38
GAA P10253 2/20 0.38
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38
HTT P42858 1/20 0.38
SIRT1 Q96EB6 1/20 0.37
TP53 P04637 2/20 0.36
POLB P06746 2/20 0.36
MAPT P10636 1/20 0.36
GRM4 Q14833 1/20 0.36
FYN P06241 2/20 0.35
LMNA P02545 1/20 0.35
NR1H4 Q96RI1 1/20 0.35
BRAF P15056 1/20 0.35
ABL1 P00519 1/20 0.35
EGFR P00533 1/20 0.35
PDGFRB P09619 1/20 0.35
BCR P11274 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7843692 0.89 TDP2 (0.40) CYP17A1TDP2KDM4ENR1H4
SCHEMBL7842830 0.89 CYP17A1 (0.41) CYP17A1TDP2ALDH1A1KDM4EMAPT
SCHEMBL7841418 0.88 CYP17A1 (0.42) CYP17A1TDP2MAPT
SCHEMBL7845051 0.86 SCN5A (0.44) CYP17A1
SCHEMBL7846790 0.85 TRPV1 (0.44) CYP17A1TDP2ALDH1A1BACE1
SCHEMBL7841770 0.84 TRPV1 (0.46) CYP17A1TDP2ALDH1A1HTTPOLB
SCHEMBL17560319 0.81 RAB9A (0.48) ALDH1A1GAAKDM4EHTTTP53
SCHEMBL7231945 0.81 BACE1 (0.37) CYP17A1TDP2ALDH1A1KDM4EHTT
SCHEMBL7843005 0.81 CYP17A1 (0.41) CYP17A1TP53POLBMAPTGRM4
SCHEMBL7846551 0.78 CNR1 (0.52) CYP17A1ALDH1A1KDM4EHTTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157022-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-28 EP disclosed
WO-2000049015-A1 PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-24 WO disclosed