SCHEMBL7844262

SCHEMBL7844262

Cc1cccc(N)c1CNC(=N)N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD44 P16070 1/20 0.39
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
HPGD P15428 3/20 0.39
CYP3A4 P08684 3/20 0.36
TDP1 Q9NUW8 1/20 0.36
TSHR P16473 1/20 0.34
PIK3CA P42336 1/20 0.34
HSD17B10 Q99714 1/20 0.33
HTT P42858 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
P2RX7 Q99572 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20957060 0.81 CYP1A2 (0.47) CD44ALDH1A1KDM4EHPGDCYP3A4
SCHEMBL2009339 0.73 CD44 (0.52) CD44ALDH1A1KDM4EHPGDCYP3A4
SCHEMBL31606366 0.73 CD44 (0.52) CD44ALDH1A1KDM4EHPGDCYP3A4
SCHEMBL4014038 0.73 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDHTTL3MBTL1
SCHEMBL19716899 0.72 HDAC1 (0.44) ALDH1A1KDM4EHPGDHSD17B10L3MBTL1
SCHEMBL7760775 0.72 CD44 (0.46) CD44ALDH1A1KDM4EHPGDCYP3A4
SCHEMBL21408116 0.71 HPGD (0.37) CD44ALDH1A1KDM4EHPGDCYP3A4
SCHEMBL3667054 0.71 CD44 (0.54) CD44ALDH1A1KDM4EHPGDCYP3A4
SCHEMBL25373683 0.71 CD44 (0.45) CD44ALDH1A1KDM4EHPGDCYP3A4
SCHEMBL2807981 0.71 SLC11A2 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1105120-A4 NON-PEPTIDE GnRH AGENTS, METHODS AND INTERMEDIATES FOR THEIR PREPARATION AGOURON PHARMA (US) 2001-12-19 EP disclosed
EP-1105120-A2 NON-PEPTIDE GnRH AGENTS, METHODS AND INTERMEDIATES FOR THEIR PREPARATION AGOURON PHARMACEUTICALS, INC. (US) 2001-06-13 EP disclosed
WO-2000020358-A2 NON-PEPTIDE GnRH AGENTS, METHODS AND INTERMEDIATES FOR THEIR PREPARATION AGOURON PHARMACEUTICALS, INC. (US) 2000-04-13 WO disclosed