SCHEMBL7844871

SCHEMBL7844871

COc1cccc2c1[C@@H]1CCNC[C@H]1CO2

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.38
SLC6A4 P31645 6/20 0.37
SLC6A2 P23975 5/20 0.37
SLC6A3 Q01959 5/20 0.37
HTR1A P08908 2/20 0.37
GNAI3 P08754 1/20 0.37
CYP2D6 P10635 1/20 0.36
CYP19A1 P11511 1/20 0.35
ADRA2C P18825 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7844867 1.00 HTR2C (0.38) HTR2CSLC6A4SLC6A2SLC6A3HTR1A
SCHEMBL6218185 0.88 CYP19A1 (0.37) HTR2CHTR1ACYP2D6CYP19A1ADRA2C
SCHEMBL6218182 0.88 CYP19A1 (0.37) HTR2CHTR1ACYP2D6CYP19A1ADRA2C
SCHEMBL7835513 0.88 CYP19A1 (0.37) HTR2CHTR1ACYP2D6CYP19A1ADRA2C
SCHEMBL7835510 0.88 CYP19A1 (0.37) HTR2CHTR1ACYP2D6CYP19A1ADRA2C
SCHEMBL6218189 0.88 CYP19A1 (0.37) HTR2CHTR1ACYP2D6CYP19A1ADRA2C
Hydrochloric Acid SCHEMBL8684946 0.86 CYP19A1 (0.36) HTR2CHTR1ACYP19A1
Hydrochloric Acid SCHEMBL8903134 0.86 CYP19A1 (0.36) HTR2CHTR1ACYP19A1
Hydrochloric Acid SCHEMBL8685813 0.86 CYP19A1 (0.36) HTR2CHTR1ACYP19A1
SCHEMBL7845327 0.80 HTR1A (0.32) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0942911-B1 BENZOPYRANOPYRROLE AND BENZOPYRANOPYRIDINE ALPHA-1 ADRENERGIC COMPOUNDS ABBOTT LAB (US) 2001-10-17 EP disclosed
US-6046207-A FOR INHIBITING ALPHA-1 ADRENORECEPTORS AND TREATING BENIGN PROSTATIC HYPERPLASIA, ALSO CALLED BENIGN PROSTATIC HYPERTROPHY, OR OTHER UROLOGICAL OR GYNECOLOGICAL DISEASES SUCH AS BLADDER OUTLET OBSTRUCTION, NEUROGENIC BLADDER ABBOTT LABORATORIES 2000-04-04 US disclosed