SCHEMBL7846462

SCHEMBL7846462

CCCCCCN1CC2C(C1)C2(C)C(c1ccccc1)S(N)(=O)=O

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 1/20 0.42
KCNH2 Q12809 2/20 0.39
PKM P14618 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
SIGMAR1 Q99720 3/20 0.37
OPRM1 P35372 3/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35
EBP Q15125 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5752500 0.69 ALDH1A1 (0.43) KCNH2ALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL20541511 0.68 HTR2A (0.43) ALDH1A1
SCHEMBL20541356 0.68 HTR2A (0.43) ALDH1A1
SCHEMBL7103282 0.68 HTR2A (0.43) ALDH1A1
SCHEMBL1837362 0.66 TP53 (0.42) SIGMAR1
SCHEMBL5757575 0.66 OPRM1 (0.50) KCNH2ALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL5754789 0.65 ALDH1A1 (0.51) KCNH2ALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL5754428 0.64 OPRM1 (0.46) OPRM1OPRD1OPRK1
SCHEMBL564038 0.64 POLB (0.43) ALDH1A1
SCHEMBL3472313 0.64 AOC3 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140828-A1 3-AZABICYCLO[3.1.0]HEXANE DERIVATIVES AS OPIATE RECEPTORS LIGANDS Pfizer Limited (GB) 2001-10-10 EP disclosed
WO-2000039089-A1 3-AZABICYCLO[3.1.0.] HEXANE DERIVATIVES AS OPIATE RECEPTORS LIGANDS PFIZER LIMITED (GB) 2000-07-06 WO disclosed