SCHEMBL7847622

SCHEMBL7847622

CC(=O)c1cc(-c2ccncc2)sc1Oc1cccc(Oc2ccc(F)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.42
GCK P35557 2/20 0.41
CYP3A4 P08684 3/20 0.40
S1PR2 O95136 1/20 0.39
RAF1 P04049 1/20 0.38
CYP1A2 P05177 3/20 0.37
CYP2C9 P11712 3/20 0.37
CYP2C19 P33261 3/20 0.37
MAPT P10636 3/20 0.37
MAPK1 P28482 2/20 0.37
MEN1 O00255 2/20 0.37
ALDH1A1 P00352 2/20 0.37
CYP2D6 P10635 2/20 0.37
HPGD P15428 2/20 0.37
KMT2A Q03164 2/20 0.37
TP53 P04637 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
ALOX12 P18054 1/20 0.37
NFKB1 P19838 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6803745 0.99 MAPK14 (0.41) MAPK14GCKCYP3A4S1PR2RAF1
SCHEMBL6801883 0.94 MAPK14 (0.46) MAPK14CYP3A4S1PR2CYP1A2CYP2C9
SCHEMBL6799622 0.87 JAK2 (0.43) MAPK14CYP3A4MAPTMAPK1MEN1
SCHEMBL6801935 0.81 MAPK1 (0.42) MAPK14GCKMAPTMAPK1MEN1
SCHEMBL6809060 0.81 MAPK14 (0.42) MAPK14MAPTMAPK1MEN1ALDH1A1
SCHEMBL6803640 0.80 MAPK1 (0.42) GCKCYP3A4S1PR2CYP1A2CYP2C9
SCHEMBL8079069 0.76 HPGD (0.38) MAPK14GCKMAPTMAPK1MEN1
SCHEMBL6803041 0.72 RAB9A (0.48) S1PR2CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL7683291 0.70 CSNK1A1 (0.60) MAPK14GCKCYP3A4CYP1A2CYP2C9
SCHEMBL17895544 0.68 MAOB (0.64) GCKCYP3A4RAF1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853083-B1 Pyridylfuran and pyridylthiophene compounds and pharmaceutical use thereof PFIZER (US) 2001-09-12 EP claimed