SCHEMBL7847878

SCHEMBL7847878

O=C(NCCN1CNc2ccc(I)cc21)C1CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.40
MTNR1A P48039 4/20 0.39
MTNR1B P49286 4/20 0.39
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
HSD17B10 Q99714 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALOX15 P16050 1/20 0.36
CASP1 P29466 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
POLB P06746 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
THRB P10828 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
SPR P35270 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6075522 0.68 MTNR1A (0.50) TSHRMTNR1AMTNR1BMEN1KMT2A
SCHEMBL12001260 0.61 ALDH1A1 (0.60) TSHRKMT2AALOX15SMN1; SMN2POLB
SCHEMBL1859048 0.61 CYP2D6 (0.52) MEN1KMT2ACYP2D6CYP2C19ALDH1A1
SCHEMBL5339230 0.60 MTNR1A (0.70) MTNR1AMTNR1B
SCHEMBL4579029 0.59
SCHEMBL14314338 0.59 MTNR1A (0.46) MTNR1AMTNR1BSMN1; SMN2SPR
SCHEMBL22071882 0.57 HSD17B10 (0.54) TSHRMEN1KMT2AHSD17B10ALOX15
SCHEMBL30799163 0.57 KMT2A (0.51) MEN1KMT2ASMN1; SMN2POLBKDM4E
SCHEMBL27383390 0.57 KMT2A (0.51) MEN1KMT2ASMN1; SMN2POLBKDM4E
SCHEMBL10050310 0.57

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077927-A1 NOVEL SUBSTITUTED CYCLIC COMPOUNDS, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ADIR ET COMPAGNIE (FR) 2001-02-28 EP disclosed
WO-1999058495-A1 NOVEL SUBSTITUTED CYCLIC COMPOUNDS, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ADIR ET COMPAGNIE (FR) 1999-11-18 WO disclosed