SCHEMBL7848321

SCHEMBL7848321

CC(=O)CCc1cc(N)n2nccc2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 6/20 0.40
CCNA1 P78396 4/20 0.40
CCNA2 P20248 2/20 0.40
CHEK1 O14757 1/20 0.40
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
CDK9 P50750 5/20 0.37
CDK7 P50613 2/20 0.37
CDK13 Q14004 1/20 0.37
CDK12 Q9NYV4 1/20 0.37
PRKAA1 Q13131 2/20 0.37
PRKAB2 O43741 1/20 0.37
PRKAG1 P54619 1/20 0.37
PRKAA2 P54646 1/20 0.37
PRKAG3 Q9UGI9 1/20 0.37
PRKAG2 Q9UGJ0 1/20 0.37
PRKAB1 Q9Y478 1/20 0.37
CCNT1 O60563 4/20 0.36
CCNH P51946 1/20 0.36
KDR P35968 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7835395 0.84 PRKAA1 (0.40) CDK2CCNA1CCNA2ADORA2AADORA1
SCHEMBL7847802 0.81 CDK9 (0.52) CDK2CCNA1CCNA2CHEK1CDK9
SCHEMBL7846977 0.77 PRKAB2 (0.48) CDK2CCNA1CCNA2CHEK1CDK9
SCHEMBL7845502 0.77 CDK2 (0.41) CDK2CCNA1CCNA2CHEK1CDK9
SCHEMBL7844352 0.75 CDK2 (0.40) CDK2CCNA1CCNA2CHEK1CDK9
SCHEMBL7847598 0.74 CDK2 (0.44) CDK2CCNA1CCNA2CHEK1CDK9
SCHEMBL7847695 0.71 CDK2 (0.39) CDK2CCNA1CCNA2CHEK1CDK9
SCHEMBL26869181 0.70 CDK2 (0.40) CDK2CCNA1CCNA2CHEK1CDK9
SCHEMBL26867731 0.70 CDK2 (0.48) CDK2CCNA1CCNA2CHEK1CDK9
SCHEMBL8180903 0.70 KDR (0.41) CDK2CCNA1CCNA2CHEK1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714898-B1 PYRAZOLO [1,5-a]PYRIMIDINE DERIVATIVE OTSUKA PHARMA CO LTD (JP) 2001-11-14 EP disclosed
US-5707997-A ANALGESICS OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1998-01-13 US disclosed
EP-0714898-A1 PYRAZOLO [1,5-a]PYRIMIDINE DERIVATIVE OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1996-06-05 EP disclosed