SCHEMBL7848569

SCHEMBL7848569

C#CC1CC[C@@H](C(N)=O)N1C(=O)[C@H](C1CC2CCC(C1)N2C(=O)N(C)C)N(C)C(=O)OC(C)(C)C

nearest known ligand 0.30

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
CHRM3 P20309 1/20 0.30
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL896326 0.76 CHRM2 (0.31) CHRM2CHRM1CHRM3
SCHEMBL7856061 0.70 DPP4 (0.41) CHRM2CHRM1CHRM3DPP4
SCHEMBL895307 0.70 DPP4 (0.41) CHRM2CHRM1CHRM3DPP4
SCHEMBL647255 0.68 DPP4 (0.41) DPP4
SCHEMBL7859357 0.68 ELANE (0.34) CHRM2CHRM1CHRM3
SCHEMBL648669 0.68 DPP4 (0.42) DPP4
SCHEMBL7856846 0.67 DPP4 (0.62) DPP4
SCHEMBL896165 0.67 DPP4 (0.62) DPP4
SCHEMBL7857237 0.67 DPP4 (0.62) DPP4
SCHEMBL3742876 0.67 ELOVL6 (0.39) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010146597-A1 2-AMINO-2- [8-(DIMETHYL CARBAMOYL)- 8-AZA- BICYCLO [3.2.1] OCT-3-YL]-EXO- ETHANOYL DERIVATIVES AS POTENT DPP-IV INHIBITORS LUPIN LIMITED (IN) 2010-12-23 WO disclosed