SCHEMBL7848865

SCHEMBL7848865

CC(C)(C)OC(=O)N1CCC(CCSc2ccc3c(c2)CCN(Cc2ccccc2)CC3)CC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 3/20 0.47
KDM4E B2RXH2 1/20 0.45
PKM P14618 1/20 0.45
PRMT5 O14744 1/20 0.45
WDR77 Q9BQA1 1/20 0.45
ACHE P22303 4/20 0.44
GPR119 Q8TDV5 3/20 0.44
BRD4 O60885 1/20 0.43
THRB P10828 2/20 0.43
GAA P10253 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
STS P08842 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
TP53 P04637 2/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7847345 0.90 ACHE (0.43) CHRM4KDM4EPKMPRMT5WDR77
SCHEMBL7849387 0.85 GPR119 (0.55) CHRM4GPR119
SCHEMBL7847536 0.84 ACHE (0.58) ACHE
SCHEMBL7847033 0.84 GPR119 (0.61) CHRM4ACHEGPR119
Hydrochloric Acid SCHEMBL7846888 0.84 ACHE (0.57) ACHE
SCHEMBL7848891 0.83 GPR119 (0.48) GPR119NPC1RAB9A
SCHEMBL7850437 0.83 GPR119 (0.46) GPR119NPC1RAB9A
SCHEMBL7855571 0.81 GPR119 (0.52) CHRM4KDM4EPKMGPR119STS
SCHEMBL7838242 0.81 CHRM4 (0.44) CHRM4KDM4EPKMPRMT5WDR77
SCHEMBL8444736 0.80 KDM4E (0.59) KDM4EPKMGPR119THRBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1122252-A1 NITROGENOUS FUSED HETEROCYCLE COMPOUNDS, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-08 EP disclosed