SCHEMBL7849348

SCHEMBL7849348

C[C@H]1C=C[C@@H](N)[C@H]2CN(c3ncc4c(=O)c(C(=O)O)cn(CCF)c4c3Cl)C[C@H]21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 5/20 0.37
LMNA P02545 3/20 0.35
CASP1 P29466 1/20 0.35
CYP2C9 P11712 2/20 0.34
CYP3A4 P08684 1/20 0.34
EPHA2 P29317 1/20 0.34
FLT4 P35916 1/20 0.34
GSK3B P49841 1/20 0.34
RARB P10826 1/20 0.34
TBXAS1 P24557 1/20 0.34
SLC6A3 Q01959 1/20 0.34
HPGD P15428 3/20 0.33
HSD17B10 Q99714 3/20 0.33
POLB P06746 2/20 0.33
XBP1 P17861 1/20 0.33
NFKB1 P19838 1/20 0.33
HTT P42858 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7849723 0.92 LMNA (0.41) KDM4EALDH1A1LMNACASP1CYP2C9
SCHEMBL7849352 0.89
SCHEMBL7851434 0.86 KDM4E (0.36) KDM4EALDH1A1LMNACASP1CYP2C9
SCHEMBL7850903 0.85 POLB (0.46) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL7851219 0.85 ALDH1A1 (0.39) KDM4EALDH1A1LMNACYP2C9CYP3A4
SCHEMBL8693387 0.85 ALDH1A1 (0.39) KDM4EALDH1A1LMNACYP2C9CYP3A4
Hydrochloric Acid SCHEMBL8697994 0.84 POLB (0.45) KDM4EALDH1A1HPGDHSD17B10POLB
Bromide SCHEMBL8692350 0.84 POLB (0.45) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL7851199 0.83 EPHA2 (0.42) KDM4EALDH1A1LMNACYP2C9CYP3A4
SCHEMBL7849726 0.81 LMNA (0.30) LMNACASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726270-B1 Derivatives of 1,6-naphthyridone carboxylic acids BAYER AG (DE) 2001-05-23 EP disclosed
EP-0726270-A1 Derivatives of 1,6-naphthyridine carboxylic acids BAYER AG (DE) 1996-08-14 EP disclosed