SCHEMBL7849445

SCHEMBL7849445

CCCCc1cc(OCCc2ccc(C(=O)O)cc2)c2ccccc2n1

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.51
KDM4E B2RXH2 1/20 0.47
CYSLTR1 Q9Y271 2/20 0.47
AGTR1 P30556 2/20 0.47
AGTR2 P50052 2/20 0.47
RARB P10826 1/20 0.46
TLR7 Q9NYK1 1/20 0.46
PTGES O14684 1/20 0.43
ALOX5 P09917 1/20 0.43
PPARG P37231 1/20 0.43
TRPV1 Q8NER1 1/20 0.43
MPL P40238 1/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8505950 0.91 TLR7 (0.49) DHODHKDM4ETLR7PTGESALOX5
SCHEMBL7838473 0.90 NR1H4 (0.49) DHODHKDM4ECYSLTR1AGTR1AGTR2
Hydrochloric Acid SCHEMBL8502040 0.89 NR1H4 (0.48) DHODHKDM4ECYSLTR1AGTR1AGTR2
SCHEMBL7839574 0.83 KDM4E (0.50) DHODHKDM4ECYSLTR1AGTR1AGTR2
SCHEMBL9182577 0.83 KDM4E (0.56) KDM4EAGTR1AGTR2
SCHEMBL8672079 0.83 KDM4E (0.53) DHODHKDM4E
Hydrochloric Acid SCHEMBL8504756 0.82 KDM4E (0.49) DHODHKDM4ECYSLTR1AGTR1AGTR2
SCHEMBL9119796 0.81 DHODH (0.53) DHODHKDM4EAGTR1AGTR2RARB
SCHEMBL7849442 0.80 RXRA (0.43) CYSLTR1PTGESALOX5PPARGPDE4A
SCHEMBL8505737 0.77 DHODH (0.55) DHODHAGTR1AGTR2PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0498723-B1 Nitrogen containing bicycle compounds, method for their preparation, their use as pharmaceutical and compositions containing them AVENTIS PHARMA SA (FR) 2001-09-19 EP disclosed
US-6004979-A ANGIOTENSIN II INHIBITORS; 4-((CARBOXY)ARYLOXY)-QUINOLINE DERIVATIVES HOECHST MARION ROUSSEL (FR) 1999-12-21 US disclosed
EP-0498723-A1 Nitrogen containing bicycle compounds, method for their preparation, their use as pharmaceutical and compositions containing them ROUSSEL UCLAF (FR) 1992-08-12 EP disclosed