SCHEMBL7849474

SCHEMBL7849474

Cc1cccc(-c2cccc3c(C(=O)Cl)cccc23)n1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.46
CCR8 P51685 1/20 0.46
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
TGFBR1 P36897 13/20 0.43
CYP2A6 P11509 1/20 0.38
HTR1A P08908 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
POLB P06746 1/20 0.37
SORT1 Q99523 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7847744 0.86 KDM4E (0.56) CCR1CCR8KDM4EALDH1A1HPGD
SCHEMBL6609571 0.78 ALDH1A1 (0.58) CCR1CCR8KDM4EALDH1A1HPGD
SCHEMBL7846725 0.78 CD38 (0.37) KDM4EALDH1A1HPGD
SCHEMBL2153429 0.75 ALDH1A1 (0.52) KDM4EALDH1A1HPGDCYP2A6
SCHEMBL12270088 0.74 CCR1 (0.58) CCR1CCR8KDM4EALDH1A1HPGD
SCHEMBL11436575 0.73 NR4A1 (0.52) KDM4EALDH1A1HPGD
SCHEMBL27887898 0.73 CDC25B (0.50) KDM4EALDH1A1HPGDHTR1AHTR1D
SCHEMBL27573254 0.71 CCR1 (0.48) CCR1CCR8KDM4EALDH1A1HPGD
SCHEMBL15945853 0.69 CCR1 (0.56) CCR1CCR8TGFBR1CYP2A6
SCHEMBL16003830 0.69 PDE10A (0.47) CCR1CCR8KDM4EALDH1A1TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140946-A2 QUINOLINE DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 2001-10-10 EP disclosed
WO-2000035919-A2 QUINOLINE DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 2000-06-22 WO disclosed