SCHEMBL7849567

SCHEMBL7849567

CC(=O)c1cc(-c2ccncc2)sc1N(C)Cc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 1/20 0.45
KDM4E B2RXH2 2/20 0.43
ABHD6 Q9BV23 1/20 0.42
POLB P06746 1/20 0.42
ROCK1 Q13464 2/20 0.42
ROCK2 O75116 1/20 0.42
JAK2 O60674 1/20 0.40
RAB9A P51151 3/20 0.40
HSD17B10 Q99714 2/20 0.40
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.39
HSD17B2 P37059 2/20 0.38
GPR142 Q7Z601 1/20 0.38
HDAC1 Q13547 2/20 0.38
GSK3B P49841 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6809616 0.99 ACKR3 (0.44) ACKR3KDM4EABHD6POLBROCK1
SCHEMBL6804230 0.77 POLB (0.44) POLBRAB9ASMN1; SMN2MAPTHPGD
SCHEMBL4918174 0.72 HSD17B2 (0.70) ACKR3HSD17B2HDAC1HDAC3HSD17B1
SCHEMBL6808781 0.70 MAPK14 (0.47) KDM4EROCK1JAK2MAPTHDAC1
SCHEMBL6799622 0.70 JAK2 (0.43) KDM4EPOLBROCK1JAK2RAB9A
SCHEMBL15263998 0.66 ABHD6 (0.69) ABHD6
SCHEMBL11331200 0.66 MAPT (0.53) ABHD6POLBALDH1A1SMN1; SMN2MAPT
SCHEMBL6799201 0.65 GABRA1 (0.36) ACKR3KDM4EABHD6POLBROCK1
SCHEMBL6801935 0.65 MAPK1 (0.42) KDM4EPOLBJAK2ALDH1A1SMN1; SMN2
SCHEMBL5182572 0.65 NR1H2 (0.50) ALDH1A1ALOX15HDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853083-B1 Pyridylfuran and pyridylthiophene compounds and pharmaceutical use thereof PFIZER (US) 2001-09-12 EP claimed