SCHEMBL7849802

SCHEMBL7849802

C1=CC(c2ccc3ccccc3c2)c2cccc3cccc1c23

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
SLC6A2 P23975 4/20 0.32
SLC6A4 P31645 6/20 0.32
SLC6A3 Q01959 3/20 0.32
CYP2D6 P10635 1/20 0.32
KCNH2 Q12809 1/20 0.32
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
TSHR P16473 2/20 0.32
HSD17B10 Q99714 2/20 0.32
TP53 P04637 1/20 0.32
MAPK1 P28482 1/20 0.32
CASP1 P29466 1/20 0.32
CASP7 P55210 1/20 0.32
HIF1A Q16665 1/20 0.32
KDM1A O60341 1/20 0.31
CYP1A1 P04798 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15814919 0.87 KDM4E (0.46) KDM4EHTR2CHTR2BSLC6A2SLC6A4
SCHEMBL28025942 0.85 KDM4E (0.45) KDM4EHTR2CHTR2BSLC6A2SLC6A4
SCHEMBL3470484 0.83 MEN1 (0.37) CYP2D6ALDH1A1HPGDTSHRHSD17B10
SCHEMBL27999787 0.82 KDM4E (0.41) KDM4EHTR2CHTR2BSLC6A2SLC6A4
SCHEMBL27862787 0.82 HTR2A (0.34) HTR2CHTR2BALDH1A1
SCHEMBL29268251 0.81 ALDH1A1 (0.32) ALDH1A1KDM1A
SCHEMBL28437775 0.81 MEN1 (0.42) SLC6A2SLC6A4SLC6A3ALDH1A1
Ethylene SCHEMBL27830648 0.81 MEN1 (0.35) ALDH1A1
SCHEMBL9473556 0.80 CA12 (0.39) MAPK1
SCHEMBL29152783 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1035848-A4 SUBSTITUTED ALKANOHYDROXAMIC ACIDS AND METHOD OF REDUCING TNF-ALPHA LEVELS CELGENE CORP (US) 2001-05-23 EP disclosed
EP-1035848-A1 SUBSTITUTED ALKANOHYDROXAMIC ACIDS AND METHOD OF REDUCING TNF-ALPHA LEVELS CELGENE CORPORATION (US) 2000-09-20 EP disclosed
WO-1999006041-A1 SUBSTITUTED ALKANOHYDROXAMIC ACIDS AND METHOD OF REDUCING TNFα LEVELS CELGENE CORPORATION (US) 1999-02-11 WO disclosed