SCHEMBL7850945

SCHEMBL7850945

Cc1ccc(C2(C)OC(=O)c3ccccc32)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 7/20 0.50
LMNA P02545 4/20 0.50
CFTR P13569 1/20 0.47
GOPC Q9HD26 1/20 0.47
MAPT P10636 4/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
POLB P06746 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
CYP3A4 P08684 3/20 0.46
GPR55 Q9Y2T6 2/20 0.46
ALDH1A1 P00352 1/20 0.46
ESR1 P03372 1/20 0.46
TP53 P04637 1/20 0.46
TYMS P04818 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
ESR2 Q92731 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11932064 0.87 CFTR (0.61) NPSR1LMNACFTRGOPCMAPT
SCHEMBL7852629 0.85 CFTR (0.46) NPSR1LMNACFTRGOPCMAPT
SCHEMBL7843306 0.85 CFTR (0.46) NPSR1LMNACFTRGOPCMAPT
SCHEMBL822834 0.81 CFTR (0.73) NPSR1LMNACFTRGOPCMAPT
SCHEMBL7855291 0.79 HSP90AA1 (0.50) NPSR1LMNACFTRGOPCMAPT
SCHEMBL19010401 0.74 CFTR (0.63) NPSR1LMNACFTRGOPCMAPT
SCHEMBL12715937 0.74 LMNA (0.85) NPSR1LMNACFTRGOPCMAPT
SCHEMBL18161910 0.72 CFTR (0.59) NPSR1LMNACFTRGOPCMAPT
SCHEMBL29672587 0.71 CFTR (0.53) NPSR1LMNACFTRGOPCMAPT
SCHEMBL361852 0.71 CFTR (0.53) NPSR1LMNACFTRGOPCMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887349-B1 Tetrahydroimidazo (2,1-a)isoquinoline derivatives AKZO NOBEL NV (NL) 2001-11-28 EP disclosed
US-5994366-A PSYCHOLOGICAL DISORDERS AKZO NOBEL NV (NL) 1999-11-30 US disclosed
EP-0887349-A1 Tetrahydroimidazo (2,1-a)isoquinoline derivatives Akzo Nobel N.V. (NL) 1998-12-30 EP disclosed