SCHEMBL7853525

SCHEMBL7853525

O=C(O)CCN1CCN(c2cc(Nc3ccc(F)c(Cl)c3)ncn2)CC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.47
EGFR P00533 13/20 0.46
ERBB3 P21860 3/20 0.46
ERBB2 P04626 3/20 0.44
ERBB4 Q15303 3/20 0.44
JAK3 P52333 1/20 0.42
AURKA O14965 1/20 0.42
AURKB Q96GD4 1/20 0.42
HPGD P15428 1/20 0.42
KMO O15229 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7853143 0.91 MCHR1 (0.43) MCHR1EGFRERBB3ERBB2ERBB4
SCHEMBL7853244 0.90 HPGD (0.48) MCHR1EGFRERBB3ERBB2ERBB4
SCHEMBL7845264 0.90 EGFR (0.47) MCHR1EGFRERBB2ERBB4JAK3
SCHEMBL7852723 0.83 EGFR (0.47) EGFRERBB3ERBB2ERBB4HPGD
SCHEMBL7852078 0.82 MALT1 (0.45) EGFRERBB3ERBB2KMO
SCHEMBL7852813 0.82 EGFR (0.42) MCHR1EGFRERBB3ERBB2ERBB4
SCHEMBL7856240 0.82 MALT1 (0.43) MCHR1EGFRERBB3ERBB2
SCHEMBL7855449 0.81 EGFR (0.46) MCHR1EGFRERBB2AURKAAURKB
SCHEMBL8630143 0.81 EGFR (0.46) EGFRERBB3ERBB2ERBB4JAK3
SCHEMBL7853953 0.79 GALR2 (0.40) EGFRERBB3ERBB2ERBB4JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1163242-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM Boehringer Ingelheim Pharma KG (DE) 2001-12-19 EP disclosed
WO-2000055162-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-21 WO disclosed