SCHEMBL7854005

SCHEMBL7854005

O=C(CN1CCC(Nc2cc(Nc3ccc(F)c(Cl)c3)ncn2)CC1)OC1CCCCC1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.46
ERBB2 P04626 3/20 0.44
EGFR P00533 11/20 0.43
S1PR1 P21453 4/20 0.42
KCNH2 Q12809 1/20 0.42
JAK3 P52333 1/20 0.40
ERBB4 Q15303 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7691002 0.89 ERBB2 (0.48) HPGDERBB2EGFRKCNH2ERBB4
SCHEMBL7853572 0.85 ERBB2 (0.44) HPGDERBB2EGFRS1PR1KCNH2
SCHEMBL7855912 0.85 ERBB2 (0.45) HPGDERBB2EGFRKCNH2ERBB4
SCHEMBL7853506 0.82 EGFR (0.46) HPGDERBB2EGFRKCNH2JAK3
SCHEMBL7574984 0.81 EGFR (0.66) HPGDERBB2EGFRJAK3ERBB4
SCHEMBL7852723 0.81 EGFR (0.47) HPGDERBB2EGFRKCNH2ERBB4
SCHEMBL7853909 0.80 EGFR (0.45) HPGDERBB2EGFRKCNH2ERBB4
SCHEMBL7852464 0.78 NOS1 (0.47) HPGDERBB2EGFRKCNH2HTT
SCHEMBL7851398 0.78 EGFR (0.50) ERBB2EGFRHTT
SCHEMBL7850948 0.77 EGFR (0.47) ERBB2EGFRJAK3HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1163242-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM Boehringer Ingelheim Pharma KG (DE) 2001-12-19 EP disclosed
WO-2000055162-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-21 WO disclosed