SCHEMBL7854068

SCHEMBL7854068

CC(C)(C)OC(=O)NC(=N)c1c(C(=O)OC(C)(C)C)[nH]c2ccc(CCNC(=O)c3cc4ccc(Cl)cc4s3)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 14/20 0.43
MAPT P10636 2/20 0.42
NAMPT P43490 1/20 0.40
F10 P00742 1/20 0.40
CNR2 P34972 1/20 0.38
PLK4 O00444 1/20 0.38
AURKA O14965 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
CHEK2 O96017 1/20 0.38
ROS1 P08922 1/20 0.38
RPS6KB1 P23443 1/20 0.38
MAPK1 P28482 1/20 0.38
FLT4 P35916 1/20 0.38
CLK2 P49760 1/20 0.38
GSK3A P49840 1/20 0.38
IRAK1 P51617 1/20 0.38
PRKX P51817 1/20 0.38
CSNK1G2 P78368 1/20 0.38
DYRK1A Q13627 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7853228 0.85 GAA (0.47) CNR1MAPTCNR2
SCHEMBL7222609 0.79 F10 (0.39) CNR1MAPTNAMPTF10PLK4
SCHEMBL7844679 0.77 MAPT (0.42) CNR1MAPTMAPK1
SCHEMBL7856628 0.77 MAPT (0.42) CNR1MAPTF10
SCHEMBL7852523 0.77 KDM4E (0.54) CNR1MAPT
SCHEMBL7852718 0.76 CA2 (0.50)
SCHEMBL7853432 0.76 CNR1 (0.44) CNR1MAPT
SCHEMBL7845669 0.76 GABRA1 (0.35) MAPT
SCHEMBL7225235 0.71 F10 (0.52) MAPTNAMPTF10PLK4AURKA
SCHEMBL7853209 0.70 HRH3 (0.36) MAPTCHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140901-A2 SUBSTITUTED (AMINOIMINOMETHYL OR AMINOMETHYL)BENZOHETEROARYL COMPOUNDS AS FACTOR XA INHIBITORS Aventis Pharmaceuticals Products Inc. (US) 2001-10-10 EP disclosed
WO-2000039087-A2 SUBSTITUTED (AMINOIMINOMETHYL OR AMINOMETHYL)BENZOHETEROARYL COMPOUNDS AS FACTOR XA INHIBITORS AVENTIS PHARMACEUTICALS PRODUCTS INC. (US) 2000-07-06 WO disclosed