SCHEMBL7855286

SCHEMBL7855286

CC1CCCN(c2ncnc3[nH]ccc23)C1.CC1CCCNC1

nearest known ligand 0.83

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 8/20 0.83
DOT1L Q8TEK3 2/20 0.63
LCK P06239 1/20 0.60
HTR2C P28335 1/20 0.54
JAK2 O60674 2/20 0.53
PRKAB2 O43741 1/20 0.52
PRKAG1 P54619 1/20 0.52
PRKAA2 P54646 1/20 0.52
PRKAA1 Q13131 1/20 0.52
PRKAG3 Q9UGI9 1/20 0.52
PRKAG2 Q9UGJ0 1/20 0.52
PRKAB1 Q9Y478 1/20 0.52
AKT2 P31751 2/20 0.52
GSK3B P49841 2/20 0.52
KIT P10721 1/20 0.52
BTK Q06187 2/20 0.52
LRRK2 Q5S007 2/20 0.50
JAK1 P23458 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20862485 0.91 JAK3 (1.00) JAK3DOT1LLCKHTR2CJAK2
SCHEMBL3954391 0.91 JAK3 (1.00) JAK3DOT1LLCKHTR2CJAK2
SCHEMBL10079358 0.84 JAK3 (1.00) JAK3DOT1LLCKHTR2CJAK2
SCHEMBL2021330 0.84 JAK3 (1.00) JAK3DOT1LLCKHTR2CJAK2
SCHEMBL7852503 0.83 DOT1L (0.66) JAK3DOT1LLCKHTR2CJAK2
SCHEMBL7850879 0.81 DOT1L (0.60) JAK3DOT1LLCKHTR2CJAK2
SCHEMBL3953791 0.80 DOT1L (0.59) JAK3DOT1LLCKHTR2CJAK2
SCHEMBL7851332 0.79 PBK (0.60) JAK3DOT1LHTR2CJAK2BTK
Nipecotic Acid SCHEMBL7851570 0.79 DOT1L (0.58) JAK3DOT1LHTR2CJAK2BTK
SCHEMBL7852777 0.78 JAK3 (0.67) JAK3DOT1LLCKHTR2CJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1087971-A1 PYRROLO 2,3-d]PYRIMIDINE COMPOUNDS Pfizer Products Inc. (US) 2001-04-04 EP disclosed
WO-1999065909-A1 PYRROLO[2,3-d]PYRIMIDINE COMPOUNDS PFIZER PRODUCTS INC. (US) 1999-12-23 WO disclosed