SCHEMBL7855396

SCHEMBL7855396

O=C(O)CCC1CCN(C2CCN(c3cc(Nc4ccc(F)c(Cl)c4)ncn3)C2)CC1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.42
MALT1 Q9UDY8 6/20 0.40
ERBB3 P21860 2/20 0.39
SCN9A Q15858 1/20 0.39
KHK P50053 1/20 0.38
DGAT1 O75907 1/20 0.38
ERBB2 P04626 1/20 0.38
MAPT P10636 1/20 0.38
FFAR4 Q5NUL3 2/20 0.37
BTK Q06187 1/20 0.37
MPL P40238 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7852078 0.82 MALT1 (0.45) EGFRMALT1ERBB3SCN9AERBB2
SCHEMBL7853143 0.82 MCHR1 (0.43) EGFRMALT1ERBB3ERBB2
SCHEMBL7590899 0.80 EGFR (0.62) EGFRERBB2MAPT
SCHEMBL7853478 0.79 BTK (0.42) EGFRMALT1ERBB3SCN9AMAPT
SCHEMBL7854432 0.79 BTK (0.45) EGFRMALT1ERBB3SCN9AMAPT
SCHEMBL7856240 0.78 MALT1 (0.43) EGFRMALT1ERBB3SCN9AERBB2
SCHEMBL8804523 0.77 EGFR (0.48) EGFRERBB3
SCHEMBL8804525 0.77 EGFR (0.48) EGFRERBB3
SCHEMBL7853525 0.77 MCHR1 (0.47) EGFRERBB3ERBB2
SCHEMBL7855000 0.75 EGFR (0.43) EGFRMALT1SCN9AERBB2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1163242-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM Boehringer Ingelheim Pharma KG (DE) 2001-12-19 EP disclosed
WO-2000055162-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-21 WO disclosed