SCHEMBL7855836

SCHEMBL7855836

O=c1c(O)c(-c2ccc3c(c2)OCO3)oc2ccc(NS(=O)(=O)c3ccc4c(c3)CNCC4)cc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.48
HTT P42858 4/20 0.48
RAB9A P51151 2/20 0.48
MEN1 O00255 2/20 0.48
TP53 P04637 2/20 0.48
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 1/20 0.48
NPC1 O15118 1/20 0.48
ALOX12 P18054 1/20 0.48
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48
PNMT P11086 2/20 0.46
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KIT P10721 1/20 0.41
PKM P14618 5/20 0.41
ALDH1A1 P00352 5/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7661345 0.89 PNMT (0.49) MAPTMEN1TP53KMT2AKDM4E
SCHEMBL7659438 0.82 GFER (0.61) MAPTHTTRAB9AMEN1TP53
SCHEMBL7664966 0.82 MAPT (0.61) MAPTHTTRAB9AMEN1TP53
SCHEMBL7665040 0.82 MAPT (0.56) MAPTHTTRAB9AMEN1TP53
SCHEMBL7657390 0.82 MAPT (0.56) MAPTHTTRAB9AMEN1TP53
SCHEMBL7654276 0.82 MAPT (0.58) MAPTHTTRAB9AMEN1TP53
SCHEMBL7858184 0.81 MAPT (0.54) MAPTHTTRAB9AMEN1TP53
SCHEMBL7659815 0.81 PKM (0.48) MAPTHTTRAB9AMEN1TP53
SCHEMBL7656710 0.80 MAPT (0.56) MAPTHTTRAB9AMEN1TP53
SCHEMBL7658164 0.80 MAPT (0.53) MAPTHTTRAB9AMEN1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109800-A1 NOVEL CDK INHIBITORS HAVING FLAVONE STRUCTURE LG CHEMICAL LIMITED (KR) 2001-06-27 EP disclosed
WO-2000012496-A1 NOVEL CDK INHIBITORS HAVING FLAVONE STRUCTURE LG CHEMICAL LTD. (KR) 2000-03-09 WO disclosed