SCHEMBL7861350

SCHEMBL7861350

CCCN(CCC)C1Cc2cc(CNS(=O)(=O)c3ccc(Cl)cc3)c(CNS(=O)(=O)c3ccc(Cl)cc3)cc2C1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.44
TSHR P16473 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
FYN P06241 1/20 0.44
DRD3 P35462 3/20 0.43
DRD2 P14416 2/20 0.43
ALDH1A1 P00352 2/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
ALOX15 P16050 1/20 0.42
MAPK1 P28482 1/20 0.42
KDM4E B2RXH2 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
TBXA2R P21731 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7854688 0.88 TBXA2R (0.54) CYP19A1DRD3DRD2ALDH1A1MAPK1
SCHEMBL7860194 0.85 CYP19A1 (0.48) CYP19A1FYNDRD3DRD2ALDH1A1
SCHEMBL7405367 0.85 MEN1 (0.42) CYP19A1TSHRNPSR1FYNDRD3
SCHEMBL7457371 0.82 DRD3 (0.61) DRD3DRD2MAPTCYP2D6TBXA2R
SCHEMBL7457363 0.82 DRD3 (0.61) DRD3DRD2MAPTCYP2D6TBXA2R
SCHEMBL8502463 0.81 DRD3 (0.50) CYP19A1DRD3DRD2ALDH1A1CYP2D6
SCHEMBL7411290 0.80 DRD3 (0.67) DRD3DRD2TBXA2R
SCHEMBL7411286 0.80 DRD3 (0.67) DRD3DRD2TBXA2R
SCHEMBL7864511 0.78 FYN (0.50) FYNDRD3DRD2ALDH1A1CYP2D6
SCHEMBL7861294 0.76 DRD3 (0.60) FYNDRD3DRD2TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0807101-B1 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS UPJOHN CO (US) 2001-06-13 EP disclosed
US-5936000-A 2-aminoindans as selective dopamine D3 ligands PHARMACIA & UPJOHN COMPANY (US) 1999-08-10 US disclosed
EP-0807101-A1 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS PHARMACIA & UPJOHN COMPANY (US) 1997-11-19 EP disclosed
WO-1996023760-A1 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS PHARMACIA & UPJOHN COMPANY (US) 1996-08-08 WO disclosed