SCHEMBL7861459

SCHEMBL7861459

C[C@@H]([C]=O)NC1CCC(C(N)c2cccnc2)CC1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
TSHR P16473 2/20 0.36
MAPT P10636 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SLC6A2 P23975 5/20 0.36
SLC6A4 P31645 5/20 0.36
ALDH1A1 P00352 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
DPP4 P27487 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35
CYP17A1 P05093 3/20 0.34
CYP19A1 P11511 3/20 0.34
SLC6A3 Q01959 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2482817 0.80 SLC6A4 (0.48) TSHRMAPTHSD17B10SLC6A2SLC6A4
Hydrochloric Acid SCHEMBL4795565 0.79 SLC6A4 (0.47) TSHRMAPTHSD17B10SLC6A2SLC6A4
SCHEMBL18228582 0.78 ALDH1A1 (0.46) TSHRALDH1A1CYP3A4CYP2D6CYP2C9
SCHEMBL19310680 0.77 SLC6A4 (0.46) KDM4ETSHRMAPTHSD17B10SLC6A2
SCHEMBL3686055 0.76 CYP11B2 (0.49) KDM4ETSHRMAPTHSD17B10SLC6A2
SCHEMBL18239433 0.75 ALDH1A1 (0.41) KDM4ETSHRMAPTHSD17B10SLC6A2
SCHEMBL3298145 0.73 SLC6A4 (0.55) SLC6A2SLC6A4CYP2D6SLC6A3
SCHEMBL6583550 0.73 GAA (0.56) KDM4ETSHRMAPTHSD17B10SLC6A2
SCHEMBL18228087 0.72 ADORA2A (0.45) TSHRALDH1A1CYP3A4CYP2D6CYP2C9
SCHEMBL18228622 0.72 SMYD3 (0.47) DPP4DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683792-B1 LHRH ANTAGONISTS HAVING MODIFIED AMINOACYL RESIDUES AT POSTIONS 5 AND 6 ABBOTT LAB (US) 2001-09-26 EP disclosed