SCHEMBL7861850

SCHEMBL7861850

O=C(CC(CCCc1ccccc1)C(=O)O)c1ccc(Br)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.53
GRIK1 P39086 1/20 0.52
HSP90AA1 P07900 2/20 0.50
MMP1 P03956 1/20 0.50
MMP2 P08253 1/20 0.50
MMP3 P08254 1/20 0.50
MMP9 P14780 1/20 0.50
MMP8 P22894 1/20 0.50
HDAC3 O15379 1/20 0.49
KMT2A Q03164 2/20 0.48
DPP4 P27487 1/20 0.48
TDP1 Q9NUW8 2/20 0.46
NPC1 O15118 1/20 0.46
CASP3 P42574 1/20 0.46
RAB9A P51151 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP3A4 P08684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7861733 0.90 TSHR (0.66) TSHRGRIK1MMP1MMP2MMP3
SCHEMBL6411354 0.87 TSHR (0.54) TSHRGRIK1MMP1MMP2MMP3
SCHEMBL12265854 0.85 KMT2A (0.59) GRIK1HSP90AA1MMP2HDAC3KMT2A
SCHEMBL8340948 0.83 TSHR (0.53) TSHRGRIK1MMP1MMP2MMP3
SCHEMBL7352438 0.83 MMP2 (0.60) TSHRGRIK1MMP1MMP2MMP3
SCHEMBL7347169 0.83 MMP2 (0.60) TSHRGRIK1MMP1MMP2MMP3
SCHEMBL7371830 0.83 MMP2 (0.60) TSHRGRIK1MMP1MMP2MMP3
SCHEMBL1857315 0.82 GRIK1 (0.57) GRIK1HSP90AA1MMP1MMP2MMP3
Bromobenzene SCHEMBL28140173 0.82 GRIK1 (0.54) GRIK1HSP90AA1MMP1MMP2MMP3
SCHEMBL5006814 0.80 KMT2A (0.48) TSHRGRIK1MMP2MMP9HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923529-B1 SUBSTITUTE 4-ARYLBUTYRIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE INHIBITORS BAYER AG (US) 2001-09-19 EP disclosed
CN-1225620-A Substituted 4-arylbutanoic acid derivatives as matrix metalloproteinase inhibitors BAYER AG (US) 1999-08-11 CN disclosed
EP-0923529-A1 SUBSITUTE 4-ARYLBUTYRIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE INHIBITORS Bayer Corporation (US) 1999-06-23 EP disclosed
US-5863915-A ENZYME INHIBITORS FOR BONES AND JOINTS BAYER CORPORATION (US) 1999-01-26 US disclosed
WO-1997043237-A1 SUBSITUTE 4-ARYLBUTYRIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE INHIBITORS BAYER CORPORATION (US) 1997-11-20 WO disclosed