SCHEMBL7862420

SCHEMBL7862420

CCCN(CCC)[C@H]1Cc2ccc(NC=O)cc2C1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 9/20 0.54
FYN P06241 1/20 0.51
ALDH1A1 P00352 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C9 P11712 1/20 0.49
ALOX15 P16050 1/20 0.49
MAPK1 P28482 1/20 0.49
DRD2 P14416 7/20 0.46
DRD4 P21917 4/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
HTR1A P08908 2/20 0.46
ADRB2 P07550 1/20 0.46
CASP1 P29466 1/20 0.46
LMNA P02545 2/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8692148 1.00 DRD3 (0.54) DRD3FYNALDH1A1CYP2D6CYP2C9
SCHEMBL9776918 0.90 DRD3 (0.61) DRD3FYNALDH1A1CYP2D6CYP2C9
SCHEMBL9441640 0.82 DRD3 (0.53) DRD3DRD2
SCHEMBL7864930 0.82 DRD3 (0.61) DRD3FYNDRD2
SCHEMBL8900096 0.82 DRD3 (0.61) DRD3FYNDRD2
SCHEMBL17822689 0.82 DRD3 (0.55) DRD3FYNALDH1A1CYP2D6CYP2C9
SCHEMBL7854607 0.78 DRD3 (0.51) DRD3FYNALDH1A1CYP2D6CYP2C9
SCHEMBL8694462 0.78 DRD3 (0.58) DRD3FYNALDH1A1CYP2D6CYP2C9
SCHEMBL8691897 0.78 DRD3 (0.54) DRD3FYNALDH1A1CYP2D6CYP2C9
SCHEMBL8690081 0.76 ALDH1A1 (0.69) ALDH1A1CYP2D6CYP2C9ALOX15MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0807101-B1 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS UPJOHN CO (US) 2001-06-13 EP disclosed
US-5936000-A 2-aminoindans as selective dopamine D3 ligands PHARMACIA & UPJOHN COMPANY (US) 1999-08-10 US disclosed
EP-0807101-A1 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS PHARMACIA & UPJOHN COMPANY (US) 1997-11-19 EP disclosed
WO-1996023760-A1 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS PHARMACIA & UPJOHN COMPANY (US) 1996-08-08 WO disclosed