SCHEMBL7862499

SCHEMBL7862499

[CH2]c1ccn(Cc2ccccc2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.49
RAB9A P51151 5/20 0.49
ALDH1A1 P00352 5/20 0.49
LMNA P02545 4/20 0.49
KDM4E B2RXH2 3/20 0.49
HPGD P15428 3/20 0.49
NFKB1 P19838 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49
CYP19A1 P11511 4/20 0.48
CACNA1G O43497 5/20 0.47
CACNA1I Q9P0X4 5/20 0.47
CACNA1H O95180 4/20 0.42
HDAC1 Q13547 3/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27724886 0.85 HDAC1 (0.50) NPC1RAB9AALDH1A1LMNAKDM4E
SCHEMBL27398369 0.78 CYP19A1 (0.50) NPC1RAB9AALDH1A1LMNAKDM4E
SCHEMBL1196571 0.77 CACNA1G (0.49) NPC1RAB9AALDH1A1KDM4ECYP19A1
SCHEMBL18577540 0.76 CYP19A1 (0.48) NPC1RAB9AALDH1A1LMNAKDM4E
SCHEMBL22149669 0.76 CYP19A1 (0.48) NPC1RAB9AALDH1A1LMNAKDM4E
SCHEMBL28260602 0.76 NPC1 (0.49) NPC1RAB9AALDH1A1LMNAKDM4E
SCHEMBL10247346 0.76 GFER (0.60) NPC1RAB9AALDH1A1LMNAKDM4E
SCHEMBL18577609 0.76 CYP19A1 (0.48) NPC1RAB9AALDH1A1LMNAKDM4E
SCHEMBL8011610 0.76 CACNA1G (0.51) NPC1RAB9AALDH1A1LMNAKDM4E
SCHEMBL634581 0.76 ALDH1A1 (0.65) NPC1RAB9AALDH1A1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107849023-A Bicyclic lactams and methods of use thereof 豪夫迈·罗氏有限公司 2018-03-27 CN disclosed
CN-101367853-A 13-membered azalides and their use as antibiotic agents PFIZER PROD INC (US) 2009-02-18 CN disclosed
EP-1131331-A1 13-MEMBERED AZALIDES AND THEIR USE AS ANTIBIOTIC AGENTS Pfizer Products Inc. (US) 2001-09-12 EP disclosed
WO-2000031097-A1 13-MEMBERED AZALIDES AND THEIR USE AS ANTIBIOTIC AGENTS PFIZER PRODUCTS INC. (US) 2000-06-02 WO disclosed