SCHEMBL7862726

SCHEMBL7862726

Cc1ccc(Cn2c(NC3CCNC(Cc4ccccc4)C3)nc3ccccc32)o1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.46
NR4A2 P43354 1/20 0.46
SSTR5 P35346 5/20 0.43
TSHR P16473 1/20 0.42
TRPC5 Q9UL62 2/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
HTT P42858 2/20 0.39
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2C9 P11712 1/20 0.37
TRPC4 Q9UBN4 1/20 0.37
MAPT P10636 2/20 0.36
HPGD P15428 1/20 0.36
MEN1 O00255 1/20 0.36
MLNR O43193 1/20 0.36
CACNA1F O60840 1/20 0.36
EED O75530 1/20 0.36
USP2 O75604 1/20 0.36
ABCB11 O95342 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864982 0.88 KCNH2 (0.45) KCNH2NR4A2SSTR5TRPC5HTT
SCHEMBL7864978 0.88 KCNH2 (0.45) KCNH2NR4A2SSTR5TRPC5HTT
SCHEMBL9697200 0.83 KCNH2 (0.62) KCNH2NR4A2SSTR5TSHRTRPC5
SCHEMBL7860380 0.82 KCNH2 (0.48) KCNH2NR4A2SSTR5TSHRTRPC5
SCHEMBL7860383 0.82 KCNH2 (0.48) KCNH2NR4A2SSTR5TSHRTRPC5
SCHEMBL7861589 0.82 KCNH2 (0.70) KCNH2NR4A2SSTR5HTTCYP1A2
SCHEMBL7861587 0.82 KCNH2 (0.70) KCNH2NR4A2SSTR5HTTCYP1A2
SCHEMBL7860295 0.81 KCNH2 (0.43) KCNH2NR4A2SSTR5NPC1RAB9A
SCHEMBL7860293 0.81 KCNH2 (0.43) KCNH2NR4A2SSTR5NPC1RAB9A
SCHEMBL7865206 0.81 KCNH2 (0.48) KCNH2NR4A2SSTR5TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869955-B1 N-ACYL-2-SUBSTITUTED-4-(BENZIMIDAZOLYL- OR IMIDAZOPYRIDINYL-SUBSTITUTED RESIDUES)-PIPERIDINES AS TACHYKININ ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2001-10-24 EP disclosed