SCHEMBL7864978

SCHEMBL7864978

Cc1ncc(Cn2c(NC3CCNC(Cc4ccccc4)C3)nc3ccccc32)o1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.45
NR4A2 P43354 2/20 0.45
SSTR5 P35346 6/20 0.42
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2C9 P11712 1/20 0.36
TRPC4 Q9UBN4 1/20 0.36
TRPC5 Q9UL62 1/20 0.36
EED O75530 2/20 0.35
MEN1 O00255 1/20 0.35
MLNR O43193 1/20 0.35
CACNA1F O60840 1/20 0.35
USP2 O75604 1/20 0.35
ABCB11 O95342 1/20 0.35
EGFR P00533 1/20 0.35
LMNA P02545 1/20 0.35
HLA-A P04439 1/20 0.35
ERBB2 P04626 1/20 0.35
TP53 P04637 1/20 0.35
LCK P06239 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864982 1.00 KCNH2 (0.45) KCNH2NR4A2SSTR5CYP1A2CYP2C19
SCHEMBL7865030 0.90 SSTR5 (0.44) KCNH2NR4A2SSTR5CYP1A2CYP2C19
SCHEMBL7865027 0.90 SSTR5 (0.44) KCNH2NR4A2SSTR5CYP1A2CYP2C19
SCHEMBL7862726 0.88 KCNH2 (0.46) KCNH2NR4A2SSTR5CYP1A2CYP2C19
SCHEMBL9303969 0.84 KCNH2 (0.60) KCNH2NR4A2SSTR5CYP1A2CYP2C19
SCHEMBL7860383 0.81 KCNH2 (0.48) KCNH2NR4A2SSTR5TRPC5MAPT
SCHEMBL7860380 0.81 KCNH2 (0.48) KCNH2NR4A2SSTR5TRPC5MAPT
SCHEMBL7861587 0.81 KCNH2 (0.70) KCNH2NR4A2SSTR5CYP1A2CYP2C19
SCHEMBL7861589 0.81 KCNH2 (0.70) KCNH2NR4A2SSTR5CYP1A2CYP2C19
SCHEMBL7860295 0.80 KCNH2 (0.43) KCNH2NR4A2SSTR5LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869955-B1 N-ACYL-2-SUBSTITUTED-4-(BENZIMIDAZOLYL- OR IMIDAZOPYRIDINYL-SUBSTITUTED RESIDUES)-PIPERIDINES AS TACHYKININ ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2001-10-24 EP disclosed